SCHEMBL178369

SCHEMBL178369

CCc1cc(O)ccc1OC

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.52
BACE1 P56817 1/20 0.49
TTR P02766 1/20 0.47
TAAR1 Q96RJ0 2/20 0.46
EGFR P00533 1/20 0.46
HSD17B10 Q99714 2/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
USP2 O75604 1/20 0.45
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
THRB P10828 1/20 0.45
ALOX15 P16050 1/20 0.45
CASP1 P29466 1/20 0.45
HTT P42858 1/20 0.45
RECQL P46063 1/20 0.45
BLM P54132 1/20 0.45
KMT2A Q03164 1/20 0.45
TDP1 Q9NUW8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29392084 0.83 MAOB (0.52) MAOBBACE1TTREGFRHSD17B10
SCHEMBL8296534 0.83 MAOB (0.57) MAOBBACE1TTRTAAR1MEN1
SCHEMBL16625523 0.83 MAOB (0.52) MAOBBACE1TTREGFRHSD17B10
SCHEMBL4847162 0.83 MAOB (0.52) MAOBBACE1TTREGFRHSD17B10
SCHEMBL8319257 0.82 MAOB (0.50) MAOBBACE1TTRTAAR1EGFR
Hydroquinone SCHEMBL9788450 0.82 MAOB (0.50) MAOBBACE1TTREGFRHSD17B10
SCHEMBL13567696 0.82 MAPT (0.47) HSD17B10KDM4EMEN1USP2ALDH1A1
SCHEMBL696593 0.81 BACE1 (0.47) MAOBBACE1TTREGFRHSD17B10
SCHEMBL4434341 0.81 BACE1 (0.48) MAOBBACE1EGFRKDM4EL3MBTL1
SCHEMBL29582819 0.81 ALOX5 (0.58) MAOBTTRMEN1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114761083-B 5-HT for treating depression 2A Agonists 罗福拉公司 2024-02-13 CN disclosed
US-20240025918-A1 KRAS G12D Inhibitors JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2024-01-25 US disclosed
EP-3962601-B1 5-HT2A AGONISTS FOR USE IN TREATMENT OF DEPRESSION Lophora ApS (DK) 2023-05-31 EP disclosed
US-11642336-B2 5-HT2A agonists for use in treatment of depression Lophora ApS (DK) 2023-05-09 US disclosed
US-11633390-B2 5-HT2A agonists for use in treatment of depression Lophora ApS (DK) 2023-04-25 US disclosed
CN-114761083-A 5-HT for the treatment of depression2AAgonists 罗福拉公司 2022-07-15 CN disclosed
US-20220062257-A1 5-HT2A AGONISTS FOR USE IN TREATMENT OF DEPRESSION Lophora ApS (DK) 2022-03-03 US disclosed
US-11246860-B2 5-HT2A agonists for use in treatment of depression Lophora ApS (DK) 2022-02-15 US disclosed
US-20210330658-A1 5-HT2A AGONISTS FOR USE IN TREATMENT OF DEPRESSION Lophora ApS (DK) 2021-10-28 US disclosed
US-20210137908-A1 5-HT2A AGONISTS FOR USE IN TREATMENT OF DEPRESSION Lophora ApS (DK) 2021-05-13 US disclosed
EP-2013176-A2 DIARYL COMPOUNDS AS NON-STEROIDAL INHIBITORS OF 17-BETA HYDROXYSTEROID DEHYDROGENASE AND/OR STEROID SULPHATASE FOR THE TREATMENT OF OESTROGEN-RELATED DISEASES SUCH AS HORMONE DEPENDENT BREAST CANCER Sterix Limited (GB) 2009-01-14 EP disclosed
EP-1881961-A1 NEW HALOALKYLSULFONE SUBSTITUTED COMPOUNDS USEFUL FOR TREATING OBESITY AND DIABETES NOVO NORDISK A/S (DK) 2008-01-30 EP disclosed
EP-1092721-B1 Chiral glucosides and their use as chiral dopants for the production of cholesteric liquid crystalline compositions BASF AG (DE) 2007-12-19 EP disclosed
WO-2007096647-A2 DIARYL COMPOUNDS AS NON-STEROIDAL INHIBITORS OF 17-BETA HYDROXYSTEROID DEHYDROGENASE AND/OR STEROID SULPHATASE FOR THE TREATMENT OF OESTROGEN-RELATED DISEASES SUCH AS HORMONE DEPENDENT BREAST CANCER STERIX LIMITED (GB) 2007-08-30 WO disclosed
US-20070037851-A1 Inhibits binding of CCR3 ligands such as eotaxins to their target cells; inhibits physiological effects of binding; therapeutic and prophylactic agents for asthma, rhinitis, dermatitis, urticaria, conjunctivitis, inflammatory bowel; tissue infiltration of eosinophils, basophils, activated T cells TEIJIN LIMITED, A JAPANESE BODY CORPORATE (JP) 2007-02-15 US disclosed
US-20070032525-A1 Piperidine derivatives having ccr3 antagonism TEIJIN LIMITED, A JAPANESE BODY CORPORATE (JP) 2007-02-08 US disclosed
WO-2006120178-A1 NEW HALOALKYLSULFONE SUBSTITUTED COMPOUNDS USEFUL FOR TREATING OBESITY AND DIABETES NOVO NORDISK A/S (DK) 2006-11-16 WO disclosed
US-4684649-A IMPROVING EFFICIENCY OF FEEDS MAROTTA ENRICO (IT) 1987-08-04 US disclosed
EP-0192992-A2 Quinoxaline derivatives useful for treatment and prophilaxis of swine dysentery and as animal growth promotants Marotta, Enrico (IT) 1986-09-03 EP disclosed
CN-86101225-A Process for the preparation of quinazoline derivatives as growth promoters for animals for the treatment and prophylaxis of swine dysentery 1986-09-03 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210330658-A1 5-HT2A AGONISTS FOR USE IN TREATMENT OF DEPRESSION HTR2A, HTR2C, HTR5A MAOB 74/4885BACE1 3577/4885TTR 4027/4885
US-20220062257-A1 5-HT2A AGONISTS FOR USE IN TREATMENT OF DEPRESSION HTR2A, HTR2C, HTR5A MAOB 74/4885BACE1 3577/4885TTR 4027/4885
US-11642336-B2 5-HT2A agonists for use in treatment of depression HTR2A, HTR2C, HTR5A MAOB 74/4885BACE1 3577/4885TTR 4027/4885
US-20070032525-A1 Piperidine derivatives having ccr3 antagonism CCR3, CCR1, CCR4 MAOB 4333/4885BACE1 4250/4885TTR 4736/4885
US-20070037851-A1 Inhibits binding of CCR3 ligands such as eotaxins to their target cells; inhibits physiological effects of binding; therapeutic and prophylactic agents for asthma, rhinitis, dermatitis, urticaria, conjunctivitis, inflammatory bowel; tissue infiltration of eosinophils, basophils, activated T cells CCR3, CCR1, CCR4 MAOB 2142/4885BACE1 3606/4885TTR 2771/4885
US-20210137908-A1 5-HT2A AGONISTS FOR USE IN TREATMENT OF DEPRESSION HTR2A, HTR2C, HTR5A MAOB 74/4885BACE1 3577/4885TTR 4027/4885
US-11633390-B2 5-HT2A agonists for use in treatment of depression HTR2A, HTR2C, HTR5A MAOB 74/4885BACE1 3577/4885TTR 4027/4885
US-11246860-B2 5-HT2A agonists for use in treatment of depression HTR2A, HTR2C, HTR5A MAOB 74/4885BACE1 3577/4885TTR 4027/4885
US-20240025918-A1 KRAS G12D Inhibitors KRAS, NRAS, HRAS MAOB 4814/4885BACE1 868/4885TTR 1672/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.