SCHEMBL17840534

SCHEMBL17840534

NCNc1nc(N)nc(-c2ccccc2)n1

nearest known ligand 0.73

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.73
ADORA2A P29274 4/20 0.60
ADORA1 P30542 3/20 0.60
ADORA3 P0DMS8 2/20 0.60
ADORA2B P29275 2/20 0.60
POLB P06746 1/20 0.60
GPR68 Q15743 5/20 0.56
HTR1A P08908 1/20 0.56
TPH1 P17752 6/20 0.52
IDH1 O75874 1/20 0.47
HSP90AA1 P07900 1/20 0.47
HSP90AB1 P08238 1/20 0.47
HTR2B P41595 1/20 0.47
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
HRH4 Q9H3N8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL197517 0.85 NPSR1 (0.71) NPSR1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL6269189 0.85 NPSR1 (0.71) NPSR1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL527618 0.82 ADORA2A (0.64) NPSR1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL8410920 0.82 NPSR1 (0.68) NPSR1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL13140029 0.82 NPSR1 (0.68) NPSR1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL11664446 0.81 NPSR1 (0.66) NPSR1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL724054 0.81 NPSR1 (0.66) NPSR1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL14058517 0.80 ADORA2A (0.67) NPSR1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL4027047 0.80 NPSR1 (0.64) NPSR1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL6975276 0.79 ADORA2A (0.60) NPSR1ADORA2AADORA1ADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9458116-B2 Benzoguanamine compound having aminomethyl group, or salt thereof, and method for manufacturing the same MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 2016-10-04 US disclosed
US-20160176827-A1 BENZOGUANAMINE COMPOUND HAVING AMINOMETHYL GROUP, OR SALT THEREOF, AND METHOD FOR MANUFACTURING THE SAME MITSUBHIS GAS CHEMICAL COMPANY, INC. (JP) 2016-06-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160176827-A1 BENZOGUANAMINE COMPOUND HAVING AMINOMETHYL GROUP, OR SALT THEREOF, AND METHOD FOR MANUFACTURING THE SAME BCAT2, GNMT, BCAT1 NPSR1 677/4885ADORA2A 2030/4885ADORA1 1503/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.