SCHEMBL17842010

SCHEMBL17842010

COc1cccc(OCCN2CCC(C(=O)NCc3ncccc3-c3ccc(Cl)cc3)CC2)c1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.50
ACKR3 P25106 2/20 0.48
DRD3 P35462 2/20 0.46
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
TSHR P16473 1/20 0.44
OPRM1 P35372 1/20 0.44
OPRD1 P41143 1/20 0.44
HRH3 Q9Y5N1 3/20 0.44
EPHX2 P34913 1/20 0.44
PKM P14618 1/20 0.43
HTR4 Q13639 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17842308 0.93 DRD2 (0.50) DRD2ACKR3DRD3SMN1; SMN2OPRM1
SCHEMBL17842183 0.82 DRD2 (0.51) DRD2OPRM1OPRD1
SCHEMBL17842566 0.77 ALDH1A1 (0.44) SMN1; SMN2
SCHEMBL23356487 0.76 DRD2 (0.83) DRD2OPRM1OPRD1
SCHEMBL17842013 0.76 DRD2 (0.83) DRD2OPRM1OPRD1
SCHEMBL23356484 0.76 DRD2 (0.83) DRD2OPRM1OPRD1
SCHEMBL17842392 0.76 CHRM1 (0.54) MAPTSMN1; SMN2
SCHEMBL17842367 0.75 SMN1; SMN2 (0.54) POLBMAPTSMN1; SMN2TSHREPHX2
SCHEMBL17842070 0.75 DRD2 (0.57) DRD2
SCHEMBL17842252 0.71 CTSD (0.39) DRD2DRD3POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233799-A1 DOPAMINE D2 RECEPTOR LIGANDS The Broad Institute Inc. (US) 2017-10-25 EP disclosed
WO-2016100823-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2016-06-23 WO disclosed