SCHEMBL17845261

SCHEMBL17845261

CCc1ccc(C(=O)NC(C)CC)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.66
RAB9A P51151 2/20 0.66
TAS1R3 Q7RTX0 1/20 0.63
TAS1R1 Q7RTX1 1/20 0.63
PLK1 P53350 1/20 0.59
LMNA P02545 1/20 0.59
HPGD P15428 3/20 0.57
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
HTT P42858 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
TDP1 Q9NUW8 1/20 0.51
KDM4E B2RXH2 1/20 0.51
MAPT P10636 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
NAMPT P43490 2/20 0.50
GAA P10253 1/20 0.50
NPC1 O15118 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
MAPK1 P28482 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19639910 1.00 ALDH1A1 (0.66) ALDH1A1RAB9ATAS1R3TAS1R1PLK1
SCHEMBL29833379 0.89 ALDH1A1 (0.66) ALDH1A1RAB9ATAS1R3TAS1R1PLK1
SCHEMBL14380335 0.85 TAS1R3 (0.67) ALDH1A1TAS1R3TAS1R1PLK1LMNA
SCHEMBL14115136 0.85 ALDH1A1 (0.70) ALDH1A1RAB9ALMNAHPGDMEN1
SCHEMBL24175853 0.84 ALDH1A1 (0.68) ALDH1A1RAB9AHPGDMEN1KMT2A
SCHEMBL15204487 0.84 ALDH1A1 (0.68) ALDH1A1RAB9AHPGDMEN1KMT2A
SCHEMBL24807877 0.83 PLK1 (0.57) ALDH1A1RAB9ATAS1R3TAS1R1PLK1
SCHEMBL24571817 0.82 ALDH1A1 (0.76) ALDH1A1RAB9ALMNAHPGDMEN1
SCHEMBL13767830 0.82 HTT (0.72) ALDH1A1RAB9ALMNAHPGDMEN1
SCHEMBL24175872 0.82 HTT (0.72) ALDH1A1RAB9ALMNAHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233836-A1 INDAZOLE SULFONAMIDE DERIVATIVES AS INVERSE AGONISTS OF RETINOID-RELATED ORPHAN RECEPTOR GAMMA (ROR GAMMA (T)) Galderma Research & Development (FR) 2017-10-25 EP disclosed
WO-2016097391-A1 INDAZOLE SULFONAMIDE DERIVATIVES AS INVERSE AGONISTS OF RETINOID-RELATED ORPHAN RECEPTOR GAMMA (ROR GAMMA (T)) GALDERMA RESEARCH & DEVELOPMENT (FR) 2016-06-23 WO disclosed