SCHEMBL17848423

SCHEMBL17848423

CC1CCCN(CCOc2ccccc2Cl)C1

nearest known ligand 0.66

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.66
KDM4E B2RXH2 9/20 0.65
GAA P10253 1/20 0.65
TDP1 Q9NUW8 1/20 0.65
HRH3 Q9Y5N1 6/20 0.59
ALDH1A1 P00352 3/20 0.58
CYP1A2 P05177 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C19 P33261 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
LMNA P02545 2/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
MEN1 O00255 1/20 0.55
PKM P14618 1/20 0.55
KMT2A Q03164 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19216371 0.85 TDP1 (0.69) KDM4EGAATDP1HRH3ALDH1A1
SCHEMBL17848522 0.84 HRH3 (0.59) KDM4EGAATDP1HRH3ALDH1A1
SCHEMBL19389876 0.81 KDM4E (0.75) KDM4EHRH3ALDH1A1LMNA
SCHEMBL9911421 0.80 TSHR (1.00) TSHRKDM4ETDP1ALDH1A1CYP1A2
SCHEMBL14970676 0.80 TSHR (1.00) TSHRKDM4ETDP1ALDH1A1CYP1A2
SCHEMBL11173592 0.80 KDM4E (0.61) KDM4EGAATDP1HRH3ALDH1A1
SCHEMBL14970552 0.79 HTT (0.64) KDM4EGAATDP1HRH3ALDH1A1
SCHEMBL19705247 0.78 HRH3 (0.83) KDM4EHRH3ALDH1A1LMNA
SCHEMBL17848619 0.77 KDM4E (0.55) KDM4EGAATDP1HRH3ALDH1A1
SCHEMBL11539872 0.74 L3MBTL1 (0.91) TSHRKDM4ETDP1ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233077-A1 DOPAMINE D2 RECEPTOR LIGANDS The Broad Institute Inc. (US) 2017-10-25 EP disclosed
WO-2016100940-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2016-06-23 WO disclosed