SCHEMBL17848433

SCHEMBL17848433

Cc1ccc(OCCN2CCC(O)CC2)c(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.49
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
DRD2 P14416 4/20 0.44
HTR1A P08908 1/20 0.44
HTR7 P34969 1/20 0.44
SYK P43405 1/20 0.44
KDM4E B2RXH2 5/20 0.43
ALDH1A1 P00352 3/20 0.43
HTT P42858 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
CRHR1 P34998 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14453570 0.86 SMN1; SMN2 (0.66) SMN1; SMN2MEN1KMT2ADRD2KDM4E
SCHEMBL19145145 0.83 SMN1; SMN2 (0.70) SMN1; SMN2MEN1KMT2ADRD2HTR1A
SCHEMBL17848636 0.82 HTR7 (0.61) DRD2HTR1AHTR7HTR2A
SCHEMBL17848328 0.79 LTA4H (0.49) DRD2HTR1AHTR7HTR2A
SCHEMBL17320456 0.76 NR1H2 (0.49) MEN1KMT2AKDM4EALDH1A1
SCHEMBL30023518 0.75 HRH1 (0.54) MEN1KMT2ADRD2KDM4EALDH1A1
SCHEMBL28870036 0.75 HRH1 (0.54) MEN1KMT2ADRD2KDM4EALDH1A1
SCHEMBL14570558 0.74 HRH3 (0.66) MEN1KMT2AALDH1A1
SCHEMBL16255800 0.74 S1PR1 (0.46) SYK
SCHEMBL12309472 0.74 MCHR1 (0.52) SMN1; SMN2MEN1KMT2AHTR1AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233077-A1 DOPAMINE D2 RECEPTOR LIGANDS The Broad Institute Inc. (US) 2017-10-25 EP disclosed
WO-2016100940-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2016-06-23 WO disclosed