SCHEMBL17848768

SCHEMBL17848768

CC1(NCc2ccc(N)cc2)CCN(C(=O)O)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPID Q08752 5/20 0.45
EPHX2 P34913 1/20 0.39
ITGB1 P05556 3/20 0.38
ITGA5 P08648 3/20 0.38
EPHX1 P07099 1/20 0.38
PTPN11 Q06124 3/20 0.38
PPIB P23284 5/20 0.37
PPIG Q13427 2/20 0.37
PPIA P62937 1/20 0.37
ITGB3 P05106 2/20 0.36
ITGAV P06756 2/20 0.36
HDAC3 O15379 2/20 0.35
HDAC4 P56524 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC7 Q8WUI4 2/20 0.35
HDAC2 Q92769 2/20 0.35
HDAC10 Q969S8 2/20 0.35
HDAC11 Q96DB2 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17262478 0.84 EPHX2 (0.43) EPHX2
SCHEMBL21855162 0.73 CASP6 (0.39) EPHX2
SCHEMBL27676112 0.72 KMT2A (0.36)
SCHEMBL17870745 0.71 CYP2C19 (0.37) EPHX2EPHX1
SCHEMBL28387866 0.70 FFAR4 (0.34) EPHX2PTPN11
SCHEMBL20766101 0.69 HDAC2 (0.51) HDAC1HDAC2
SCHEMBL17262465 0.69 RORC (0.47) HDAC1
SCHEMBL17848769 0.69 CASP6 (0.36) PPIDPPIB
SCHEMBL19641201 0.69 ALDH1A1 (0.48)
SCHEMBL18154336 0.69 ALDH1A1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233077-A1 DOPAMINE D2 RECEPTOR LIGANDS The Broad Institute Inc. (US) 2017-10-25 EP disclosed
WO-2016100940-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2016-06-23 WO disclosed