SCHEMBL17848770

SCHEMBL17848770

CC1(Oc2ccccc2Cl)CCN(CCOc2ccc(F)cc2)CC1

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 16/20 0.67
TSHR P16473 1/20 0.49
LTA4H P09960 1/20 0.49
HTR1A P08908 1/20 0.47
DRD1 P21728 1/20 0.47
DRD5 P21918 1/20 0.47
SLC6A2 P23975 1/20 0.47
HTR2A P28223 1/20 0.47
SLC6A4 P31645 1/20 0.47
HTR7 P34969 1/20 0.47
HRH1 P35367 1/20 0.47
DRD3 P35462 1/20 0.47
HTR2B P41595 1/20 0.47
USP2 O75604 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17848775 0.92 DRD2 (0.80) DRD2TSHRLTA4H
SCHEMBL17848380 0.87 DRD2 (0.80) DRD2LTA4HHTR1ADRD1DRD5
SCHEMBL17848502 0.85 DRD2 (0.76) DRD2TSHR
SCHEMBL17848766 0.85 DRD2 (0.65) DRD2ALDH1A1
SCHEMBL17848429 0.85 DRD2 (0.77) DRD2TSHR
SCHEMBL17848317 0.84 DRD2 (0.72) DRD2TSHRHTR1AHTR7ALDH1A1
SCHEMBL17848339 0.82 DRD2 (0.80) DRD2TSHRLTA4HHTR1AHTR7
SCHEMBL17848595 0.81 DRD2 (0.78) DRD2LTA4HHTR1AHTR2AHRH1
SCHEMBL17848571 0.81 DRD2 (1.00) DRD2LTA4HALDH1A1
SCHEMBL17848350 0.81 DRD2 (0.77) DRD2HTR1ADRD1DRD5SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233077-A1 DOPAMINE D2 RECEPTOR LIGANDS The Broad Institute Inc. (US) 2017-10-25 EP disclosed
WO-2016100940-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2016-06-23 WO disclosed