SCHEMBL17849217

SCHEMBL17849217

N=C(c1ccc(N2CCSCC2)cc1)c1c(Nc2c(F)cccc2F)c(Cl)c[nH]c1=O

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.33
EGFR P00533 2/20 0.31
ROCK1 Q13464 2/20 0.31
AKR1C3 P42330 1/20 0.31
NTRK1 P04629 1/20 0.31
MAPK7 Q13164 1/20 0.31
F10 P00742 1/20 0.31
MAPT P10636 2/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPK1 P28482 1/20 0.30
MPI P34949 1/20 0.30
KMT2A Q03164 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
JAK2 O60674 1/20 0.30
JAK1 P23458 1/20 0.30
TYK2 P29597 1/20 0.30
JAK3 P52333 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623587 0.90 ROCK1 (0.39) DGAT1ROCK1NTRK1MAPK7MAPT
SCHEMBL17849203 0.88 ROCK1 (0.40) DGAT1ROCK1NTRK1MAPK7MAPT
SCHEMBL17849212 0.83 ITGB3 (0.37) F10MEN1KMT2A
SCHEMBL17849193 0.82 F10 (0.43) F10MAPTALDH1A1
SCHEMBL17849189 0.80 RAB9A (0.45) NTRK1KDM4EALDH1A1
SCHEMBL17849207 0.80 ROCK1 (0.39) ROCK1NTRK1MAPK7MAPTKDM4E
SCHEMBL17849219 0.80 RAF1 (0.42) ROCK1NTRK1MAPTKDM4EMEN1
SCHEMBL17849202 0.80 SMN1; SMN2 (0.44) MAPK7MAPTKDM4EMEN1ALDH1A1
SCHEMBL17849208 0.78 HDAC6 (0.33) MAPTALDH1A1KMT2A
SCHEMBL17849214 0.78 TYK2 (0.38) ROCK1MAPTKDM4EALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed