SCHEMBL17849189

SCHEMBL17849189

N=C(c1ccc(CN2CCOCC2)cc1)c1c(Nc2c(F)cccc2F)c(Cl)c[nH]c1=O

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.45
LMNA P02545 1/20 0.45
NPC1 O15118 5/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
TP53 P04637 2/20 0.42
CYP2A13 Q16696 1/20 0.42
ALDH1A1 P00352 2/20 0.41
NTRK1 P04629 1/20 0.41
HIF1A Q16665 3/20 0.40
EPAS1 Q99814 3/20 0.40
HRH3 Q9Y5N1 1/20 0.38
HPGD P15428 1/20 0.38
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17849200 0.87 CYP2A13 (0.39) RAB9ALMNANPC1SMN1; SMN2TP53
SCHEMBL17849190 0.86 LTA4H (0.33) RAB9ALMNAALDH1A1NTRK1
SCHEMBL17849203 0.85 ROCK1 (0.40) RAB9ANPC1ALDH1A1NTRK1HPGD
SCHEMBL17849208 0.85 HDAC6 (0.33) LMNASMN1; SMN2TP53ALDH1A1
SCHEMBL17849211 0.84 L3MBTL1 (0.38) RAB9ASMN1; SMN2ALDH1A1NTRK1HRH3
SCHEMBL17849202 0.83 SMN1; SMN2 (0.44) RAB9ALMNANPC1SMN1; SMN2TP53
SCHEMBL16726665 0.82 ALDH2 (0.33)
SCHEMBL16623450 0.81 NPC1 (0.32) LMNANPC1
SCHEMBL17849217 0.80 DGAT1 (0.33) ALDH1A1NTRK1KDM4E
SCHEMBL17849197 0.79 ALDH1A1 (0.38) RAB9ALMNANPC1SMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed