SCHEMBL17849245

SCHEMBL17849245

N#Cc1cccc(F)c1Nc1cc[nH]c(=O)c1C(=N)c1ccc(N2CCOCC2)nc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
CNR2 P34972 1/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
JAK2 O60674 3/20 0.38
TYK2 P29597 3/20 0.38
KCNQ3 O43525 1/20 0.37
KCNQ2 O43526 1/20 0.37
ALDH1A1 P00352 2/20 0.37
USP30 Q70CQ3 1/20 0.37
EGLN1 Q9GZT9 3/20 0.36
DGAT1 O75907 1/20 0.36
EGFR P00533 1/20 0.36
LRRK2 Q5S007 1/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623509 0.92 NPC1 (0.46) NPC1RAB9ACNR2KCNQ3KCNQ2
SCHEMBL17849244 0.89 TYK2 (0.40) JAK2TYK2ALDH1A1EGFRLRRK2
SCHEMBL17849188 0.80 EGFR (0.40) NPC1RAB9AJAK2ALDH1A1DGAT1
SCHEMBL17849246 0.76 PARP1 (0.34) JAK2TYK2LRRK2
SCHEMBL17849222 0.75 ALDH1A1 (0.36) NPC1RAB9AGAATYK2ALDH1A1
SCHEMBL17849216 0.75 AR (0.33) NPC1RAB9AEGFRAKT1
SCHEMBL17849214 0.72 TYK2 (0.38) NPC1RAB9ATSHRJAK2TYK2
SCHEMBL17849247 0.72 MAPT (0.41) NPC1RAB9AGAAALDH1A1EGFR
SCHEMBL16623493 0.71 TYK2 (0.39) JAK2TYK2
SCHEMBL17849249 0.71 EGFR (0.40) TSHRJAK2ALDH1A1EGFRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed