SCHEMBL17849249

SCHEMBL17849249

N=C(c1ccc(N2CCNCC2)cc1)c1c(Nc2c(F)cccc2F)cc[nH]c1=O

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGFR P00533 14/20 0.40
ALDH1A1 P00352 2/20 0.39
USP2 O75604 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
KDR P35968 1/20 0.38
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
MAOB P27338 1/20 0.36
WEE1 P30291 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17849188 0.90 EGFR (0.40) EGFRALDH1A1JAK2JAK1MAOB
SCHEMBL16623503 0.87 EGFR (0.35) EGFRJAK2JAK1
SCHEMBL17849221 0.85 EIF2AK2 (0.34) EGFRJAK2JAK1
SCHEMBL17849248 0.85 EGFR (0.41) EGFRALDH1A1JAK2JAK1
SCHEMBL16623568 0.84 EGFR (0.38) EGFRJAK2JAK1
SCHEMBL16623565 0.82 ALDH1A1 (0.41) ALDH1A1TSHR
SCHEMBL17849244 0.82 TYK2 (0.40) EGFRALDH1A1HSD17B10JAK2JAK1
SCHEMBL18052623 0.82 EGFR (0.36) EGFRKDRJAK2JAK1
SCHEMBL17849247 0.81 MAPT (0.41) EGFRALDH1A1MAOB
SCHEMBL16623558 0.81 PARP1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed