SCHEMBL17849533

SCHEMBL17849533

CC1CN(C(=O)c2ccc(N)c(Cl)c2)C1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.56
HPGD P15428 4/20 0.46
ALDH1A1 P00352 3/20 0.46
POLB P06746 1/20 0.46
PLA2G1B P04054 1/20 0.46
ATG4B Q9Y4P1 1/20 0.46
GAA P10253 1/20 0.45
PDK2 Q15119 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PKM P14618 1/20 0.43
HSD11B1 P28845 4/20 0.43
KMT2A Q03164 1/20 0.43
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12525209 0.84 LRRK2 (0.53) LRRK2HPGDALDH1A1POLBPDK2
SCHEMBL22012072 0.82 HDAC1 (0.47) HPGDALDH1A1PLA2G1BATG4BGAA
SCHEMBL3454797 0.80 HPGD (0.59) LRRK2HPGDALDH1A1POLBPLA2G1B
SCHEMBL12526825 0.80 LRRK2 (0.68) LRRK2HPGDALDH1A1HSD17B10PKM
SCHEMBL11293154 0.80 HPGD (0.73) LRRK2HPGDALDH1A1POLBPKM
SCHEMBL21938853 0.79 HSD11B1 (0.50) LRRK2HPGDALDH1A1POLBPLA2G1B
SCHEMBL12525213 0.79 POLB (0.62) LRRK2HPGDALDH1A1POLBPKM
SCHEMBL15653084 0.78 LRRK2 (0.63) LRRK2HPGDHSD17B10PKMHSD11B1
SCHEMBL15653083 0.78 LRRK2 (0.63) LRRK2HPGDHSD17B10PKMHSD11B1
SCHEMBL15172215 0.78 GAA (0.55) LRRK2HPGDALDH1A1POLBPLA2G1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371319-B2 Pyrrolopyridineamino derivatives as MPS1 inhibitors CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2016-06-21 US disclosed