SCHEMBL17850388

SCHEMBL17850388

Cc1ccc(C(=O)Nc2cnn(CCN3CCOCC3)c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KA2 Q15349 1/20 0.56
MAPK1 P28482 2/20 0.55
NPC1 O15118 2/20 0.55
RAB9A P51151 2/20 0.55
TP53 P04637 1/20 0.55
PKM P14618 1/20 0.55
CYP2C19 P33261 2/20 0.55
CYP1A2 P05177 1/20 0.55
MAPT P10636 1/20 0.55
LMNA P02545 2/20 0.53
HTT P42858 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.52
GAA P10253 2/20 0.52
ALDH1A1 P00352 1/20 0.52
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
TSHR P16473 2/20 0.50
CYP3A4 P08684 1/20 0.50
EGFR P00533 1/20 0.49
KDR P35968 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15317700 0.89 MAPT (0.57) RPS6KA2MAPK1NPC1RAB9AMAPT
SCHEMBL3258508 0.83 RPS6KA2 (0.48) RPS6KA2RAB9ATP53CYP2C19LMNA
SCHEMBL10195016 0.76 TAS2R8 (0.53) RPS6KA2NPC1RAB9ALMNASMN1; SMN2
SCHEMBL14409565 0.75 RAB9A (0.79) MAPK1NPC1RAB9ATP53PKM
SCHEMBL8178868 0.75 TAS2R8 (0.43) RPS6KA2MAPK1KDRIKBKETBK1
SCHEMBL763452 0.74 HTT (0.78) MAPK1CYP2C19LMNAHTTSMN1; SMN2
SCHEMBL280240 0.74 MEN1 (0.76) MAPK1CYP2C19LMNAHTTALDH1A1
SCHEMBL15214859 0.74 MAP4K4 (0.50) MAPK1NPC1RAB9ALMNASMN1; SMN2
Hydrochloric Acid SCHEMBL3257525 0.73 TAS2R8 (0.43) RPS6KA2MAPK1KDRIKBKETBK1
SCHEMBL6937374 0.73 JAK2 (0.41) MAPK1RAB9AMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655357-B1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO SA (CH) 2016-06-22 EP disclosed