SCHEMBL178526

SCHEMBL178526

CC(C)c1cccc(NC(=O)N2CCOCC2)c1

nearest known ligand 0.71

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.71
RAB9A P51151 3/20 0.71
CYP2C9 P11712 1/20 0.62
CYP2C19 P33261 1/20 0.62
NPY5R Q15761 3/20 0.59
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
GAA P10253 2/20 0.57
MAPT P10636 1/20 0.57
HPGD P15428 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
TRPV1 Q8NER1 1/20 0.54
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL178415 0.85 KDM4E (0.65) NPC1RAB9ACYP2C9CYP2C19MEN1
SCHEMBL2399070 0.84 POLB (0.61) NPC1RAB9ACYP2C9CYP2C19MEN1
SCHEMBL104586 0.83 RAB9A (1.00) NPC1RAB9ACYP2C9CYP2C19MEN1
SCHEMBL12693 0.82 ALDH1A1 (0.76) NPC1RAB9ACYP2C9CYP2C19MEN1
SCHEMBL19016264 0.81 ALDH1A1 (0.67) MEN1KMT2ASMN1; SMN2GAANPSR1
SCHEMBL15033571 0.80 NPC1 (0.70) NPC1RAB9ACYP2C9CYP2C19MEN1
SCHEMBL21348459 0.80 NPC1 (0.65) NPC1RAB9ACYP2C9CYP2C19NPY5R
SCHEMBL1097789 0.79 NPC1 (0.68) NPC1RAB9ACYP2C9CYP2C19MEN1
SCHEMBL1407210 0.79 NPC1 (0.68) NPC1RAB9ACYP2C9CYP2C19MEN1
SCHEMBL20237020 0.79 SMN1; SMN2 (0.68) NPC1RAB9ACYP2C9CYP2C19NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120059162-A1 FUSED IMIDAZOLE DERIVATIVE HAVING TTK INHIBITORY ACTION ONCOTHERAPY SCIENCE, INC. (JP) 2012-03-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120059162-A1 FUSED IMIDAZOLE DERIVATIVE HAVING TTK INHIBITORY ACTION NR0B1, GRK7, NR5A2 NPC1 1892/4885RAB9A 3030/4885CYP2C9 3302/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.