SCHEMBL17858535

SCHEMBL17858535

C=CC(c1cccc(OC)c1)c1ccccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
NFE2L2 Q16236 1/20 0.40
DRD2 P14416 2/20 0.40
OPRD1 P41143 1/20 0.40
VDR P11473 1/20 0.40
P4HB P07237 1/20 0.39
GRM5 P41594 2/20 0.39
GRM4 Q14833 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
CASR P41180 1/20 0.38
SLC10A1 Q14973 1/20 0.38
AHR P35869 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
NPC1 O15118 1/20 0.37
PKM P14618 1/20 0.37
RAB9A P51151 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29029215 0.78 SLC6A2 (0.57) OPRD1SLC6A2SLC6A4SLC6A3SLC10A1
SCHEMBL10569701 0.78 SLC6A2 (0.57) OPRD1SLC6A2SLC6A4SLC6A3SLC10A1
SCHEMBL17842030 0.78 DYRK1A (0.45) DYRK1ACLK4DRD2VDRP4HB
SCHEMBL30638827 0.78 SLC6A3 (0.64) DYRK1ACLK4NFE2L2DRD2VDR
SCHEMBL30879872 0.78 DYRK1A (0.45) DYRK1ACLK4DRD2VDRP4HB
SCHEMBL29518433 0.78 DYRK1A (0.45) DYRK1ACLK4NFE2L2DRD2VDR
SCHEMBL28557150 0.78 SLC6A3 (0.64) DYRK1ACLK4NFE2L2DRD2VDR
SCHEMBL17842130 0.78 DYRK1A (0.45) DYRK1ACLK4NFE2L2DRD2VDR
Hydrochloric Acid SCHEMBL17842300 0.77 ROCK1 (0.44) DYRK1ACLK4DRD2VDRP4HB
SCHEMBL29588451 0.77 DYRK1A (0.44) DYRK1ACLK4NFE2L2DRD2VDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016100823-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2016-06-23 WO disclosed