SCHEMBL17860701

SCHEMBL17860701

Clc1cccc(-c2ccc(I)cn2)c1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.54
MAOB P27338 1/20 0.54
IDO1 P14902 4/20 0.49
MAP4K4 O95819 2/20 0.43
KMO O15229 2/20 0.43
FYN P06241 1/20 0.43
HSD17B1 P14061 1/20 0.42
HSD17B2 P37059 1/20 0.42
CYP19A1 P11511 1/20 0.42
GRM5 P41594 1/20 0.41
DHFR P00374 1/20 0.41
SCN2A Q99250 1/20 0.41
NOTUM Q6P988 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2134773 0.79 KDM1A (0.61) KDM1AMAOBIDO1MAP4K4KMO
SCHEMBL31689000 0.79 KDM1A (0.54) KDM1AMAOBIDO1MAP4K4KMO
SCHEMBL10264655 0.79 CYP3A4 (0.54) KDM1AMAOBIDO1MAP4K4KMO
SCHEMBL6863681 0.79 HPGDS (0.56) IDO1MAP4K4KMOFYNHSD17B1
SCHEMBL19992669 0.77 KDM1A (0.49) KDM1AMAOBKMOFYNNOTUM
SCHEMBL15097694 0.77 LDHA (0.52)
SCHEMBL2609359 0.75 MAOB (0.50) KDM1AMAOBIDO1MAP4K4KMO
SCHEMBL19992829 0.75 KDM1A (0.57) KDM1AMAOBIDO1KMOSCN2A
SCHEMBL17882026 0.75 MAOB (0.50) KDM1AMAOBIDO1FYNDHFR
SCHEMBL11683554 0.74 KDM1A (0.53) KDM1AMAOBIDO1MAP4K4KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016100578-A2 ANTIMICROBIAL POLYMYXINS FOR TREATMENT OF BACTERIAL INFECTIONS MICURX PHARMACEUTICALS, INC. (US) 2016-06-23 WO disclosed