SCHEMBL17864631

SCHEMBL17864631

Cc1cc(C)c2cc(C(=O)OC(C)(C)C)oc2c1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA9 Q16790 1/20 0.36
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
KDM4E B2RXH2 3/20 0.34
HSD17B10 Q99714 3/20 0.34
HPGD P15428 2/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TSHR P16473 1/20 0.34
THRB P10828 2/20 0.33
MAPT P10636 1/20 0.33
UBE2N P61088 1/20 0.33
TP53 P04637 1/20 0.33
MCL1 Q07820 1/20 0.33
AR P10275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17864553 0.83 RARA (0.39) CA12CA1CA9CYP2C9CYP2C19
SCHEMBL29394908 0.83 RARA (0.39) CA12CA1CA9CYP2C9CYP2C19
SCHEMBL17864632 0.77 MCL1 (0.46) L3MBTL1KDM4EHSD17B10HPGDKMT2A
SCHEMBL23691678 0.70 RARA (0.36) THRBMAPTTP53
SCHEMBL12867871 0.70 MAPT (0.38) CA12CA1CA9CYP2C9CYP2C19
SCHEMBL19583312 0.68 CISD2 (0.35) L3MBTL1THRBMAPTTP53AR
SCHEMBL22835128 0.67 HDAC4 (0.44) CA12CA1CA9CYP2C19NPSR1
SCHEMBL5655693 0.66 KDM4E (0.45) CA12CA1CA9NPSR1L3MBTL1
SCHEMBL3977133 0.66 CHRNA4 (0.38) CA12CA1CA9CYP2C9CYP2C19
SCHEMBL17864589 0.65 CA12 (0.40) CA12CA1CA9CYP2C19KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016097004-A1 BICYCLOHETEROARYL-HETEROARYL-BENZOIC ACID COMPOUNDS AS RETINOIC ACID RECEPTOR BETA (RARβ) AGONISTS KING'S COLLEGE LONDON (GB) 2016-06-23 WO disclosed