SCHEMBL17864752

SCHEMBL17864752

CCCCOc1cc(Br)c(C)cc1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.47
PDE3A Q14432 1/20 0.47
L3MBTL1 Q9Y468 6/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
MAPT P10636 6/20 0.44
HPGD P15428 3/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
TSHR P16473 1/20 0.44
TDP1 Q9NUW8 2/20 0.42
LMNA P02545 2/20 0.41
TP53 P04637 1/20 0.41
SMPD1 P17405 3/20 0.40
PTPN1 P18031 2/20 0.40
MAPK1 P28482 1/20 0.40
KDM4E B2RXH2 1/20 0.40
PDE4B Q07343 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17529471 1.00 PDE3B (0.47) PDE3BPDE3AL3MBTL1SMN1; SMN2MAPT
SCHEMBL3370500 0.86 L3MBTL1 (0.48) L3MBTL1SMN1; SMN2MAPTHPGDNPC1
SCHEMBL5843168 0.86 THRA (0.43) SMN1; SMN2SMPD1
SCHEMBL21823607 0.84 LMNA (0.49) PDE3BPDE3AL3MBTL1SMN1; SMN2MAPT
SCHEMBL31096332 0.84 LMNA (0.49) PDE3BPDE3AL3MBTL1SMN1; SMN2MAPT
SCHEMBL15691067 0.82 PDE3B (0.48) PDE3BPDE3AL3MBTL1SMN1; SMN2MAPT
SCHEMBL15839257 0.81 L3MBTL1 (0.47) PDE3BPDE3AL3MBTL1SMN1; SMN2MAPT
SCHEMBL18466878 0.81 PDE3B (0.43) PDE3BPDE3AL3MBTL1SMN1; SMN2MAPT
SCHEMBL29622968 0.81 CYP1A2 (0.45) L3MBTL1SMN1; SMN2MAPTHPGDNPC1
SCHEMBL7739532 0.81 CYP1A2 (0.45) L3MBTL1SMN1; SMN2MAPTHPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016100391-A1 2-PHENETHENYLTETRAHYDRO ISOQUINOLINES USEFUL AS ANTI-HIV COMPOUNDS Prosetta Antiviral, Inc. (US) 2016-06-23 WO disclosed