SCHEMBL17865487

SCHEMBL17865487

C=CCC(C(=O)c1cc(F)ccc1F)N(C(=O)O)C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.40
CES1 P23141 2/20 0.40
MDM2 Q00987 11/20 0.36
RIPK1 Q13546 2/20 0.33
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
MEN1 O00255 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
PSMB11 A5LHX3 1/20 0.31
PSMA7 O14818 1/20 0.31
PSMB1 P20618 1/20 0.31
PSMA1 P25786 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17102154 0.81 CES2 (0.40) CES2CES1MDM2RIPK1
SCHEMBL17865488 0.78 MDM2 (0.40) CES2CES1MDM2PSMB5
SCHEMBL17865486 0.71 CES2 (0.44) CES2CES1MDM2PSMB11PSMA7
SCHEMBL17102140 0.70 CTSS (0.43) CES2CES1HPGD
SCHEMBL17121664 0.69 CES2 (0.46) CES2CES1MDM2PSMB11PSMA7
SCHEMBL1665547 0.69
SCHEMBL4149785 0.69 GRIK1 (0.33)
SCHEMBL1665550 0.69
SCHEMBL21838666 0.66
SCHEMBL15561658 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2997008-B1 PROCESS FOR THE PREPARATION OF KEY INTERMEDIATES OF OMARIGLIPTIN ITALIANA SINT SPA (IT) 2016-06-29 EP claimed