SCHEMBL17865488

SCHEMBL17865488

C=CCC(C(=O)c1cc(F)ccc1F)N(Cc1ccccc1)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 10/20 0.40
CES2 O00748 2/20 0.39
CES1 P23141 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
POLB P06746 1/20 0.35
DPP4 P27487 1/20 0.35
DPP9 Q86TI2 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
PSMB5 P28074 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17865487 0.78 CES2 (0.40) MDM2CES2CES1PSMB5
SCHEMBL17102165 0.71 CASP3 (0.47)
SCHEMBL17865486 0.70 CES2 (0.44) MDM2CES2CES1PSMB5
SCHEMBL17121664 0.69 CES2 (0.46) MDM2CES2CES1PSMB5
SCHEMBL5514599 0.68 NFE2L2 (0.43) TDP1DPP4DPP9DPP7
SCHEMBL5514603 0.68 NFE2L2 (0.43) TDP1DPP4DPP9DPP7
SCHEMBL22654029 0.67 CYP2C19 (0.49) L3MBTL1TDP1POLB
SCHEMBL924474 0.64 CYP2C19 (0.46) L3MBTL1POLB
SCHEMBL8079850 0.64 MEN1 (0.48) L3MBTL1POLB
SCHEMBL8966854 0.64 MEN1 (0.48) L3MBTL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2997008-B1 PROCESS FOR THE PREPARATION OF KEY INTERMEDIATES OF OMARIGLIPTIN ITALIANA SINT SPA (IT) 2016-06-29 EP claimed