SCHEMBL17865944

SCHEMBL17865944

CN([C@H]1C[C@@H](n2ccc3c(NCc4ccc5c(c4)OCO5)ncnc32)C[C@@H]1O)S(=O)(=O)O

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 14/20 0.49
KDM4E B2RXH2 4/20 0.49
MAPT P10636 4/20 0.49
ALDH1A1 P00352 4/20 0.49
TSHR P16473 3/20 0.49
HSD17B10 Q99714 3/20 0.49
HPGD P15428 2/20 0.49
NPSR1 Q6W5P4 2/20 0.49
RXFP1 Q9HBX9 2/20 0.49
MAPK1 P28482 3/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
EGFR P00533 1/20 0.47
AURKA O14965 1/20 0.44
RPS6KB1 P23443 1/20 0.44
AURKB Q96GD4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17865976 0.86 CCNA2 (0.44) AURKARPS6KB1
SCHEMBL17865956 0.86 NAE1 (0.43) KDM4EMAPTALDH1A1TSHRHSD17B10
SCHEMBL17865942 0.85 KDM4E (0.48) PDE5AKDM4EMAPTALDH1A1TSHR
SCHEMBL17865921 0.85 METTL3 (0.54) PDE5AMAPTMAPK1
SCHEMBL17865958 0.85 TP53 (0.45) MAPTRXFP1MAPK1EGFR
SCHEMBL17866025 0.84 KDM4E (0.53) PDE5AKDM4EMAPTALDH1A1TSHR
SCHEMBL17865924 0.82 UBA6 (0.38)
SCHEMBL192776 0.82 NAE1 (0.57) PDE5AKDM4EMAPTALDH1A1TSHR
SCHEMBL17865917 0.81 UBA6 (0.42)
SCHEMBL17865973 0.81 UBA6 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2402334-B1 Inhibitors of E1 Activating Enzymes MILLENNIUM PHARM INC (US) 2016-06-29 EP claimed