SCHEMBL1786889

SCHEMBL1786889

Clc1ccc2c(c1)C=CC2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.38
HTR2A P28223 2/20 0.38
HTR2B P41595 1/20 0.38
PNMT P11086 1/20 0.35
CMA1 P23946 1/20 0.34
AHR P35869 1/20 0.34
METAP1 P53582 1/20 0.33
TP53 P04637 1/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
F7 P08709 1/20 0.32
PARP1 P09874 1/20 0.32
F3 P13726 1/20 0.32
PARP10 Q53GL7 1/20 0.32
HSD17B3 P37058 1/20 0.32
KDM1A O60341 1/20 0.32
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31513977 0.82 HTR2C (0.38) HTR2CHTR2AHTR2BPNMTAHR
SCHEMBL1896564 0.82 HTR2C (0.38) HTR2CHTR2AHTR2BPNMTAHR
SCHEMBL6832707 0.78 HTR2A (0.35) HTR2CHTR2AHTR2BPNMTCMA1
SCHEMBL924413 0.77 CYP1A2 (0.35) HTR2BMETAP1TP53CA1CA2
SCHEMBL9629684 0.76 CA1 (0.34) CA1CA2
SCHEMBL275807 0.74 CA1 (0.33) CA1CA2
SCHEMBL3755892 0.74 ESR1 (0.38) HTR2CHTR2AHTR2BCYP3A4ALOX15
SCHEMBL2730845 0.73 MAPT (0.36) CA1CA2CYP3A4SMN1; SMN2MEN1
SCHEMBL2965930 0.73 TRPA1 (0.37) HTR2CHTR2AHTR2BPNMTCMA1
SCHEMBL275808 0.73 PBRM1 (0.36) CA1CA2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 46 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060052620-A1 Preparation of substituted indenes BASELL POLYOLEFINE GMBH (DE) 2006-03-09 US claimed
CN-1653021-A Preparation of substituted indenes BASELL POLYOLEFINE GMBH (DE) 2005-08-10 CN claimed
EP-1492749-A1 PREPARATION OF SUBSTITUTED INDENES Basell Polyolefine GmbH (DE) 2005-01-05 EP claimed
WO-2003084904-A1 PREPARATION OF SUBSTITUTED INDENES BASELL POLYOLEFINE GMBH (DE) 2003-10-16 WO claimed
EP-4392410-A1 TRANSCRIPTION FACTOR BRN2 INHIBITORY COMPOUNDS FOR USE AS THERAPEUTICS The University of British Columbia (CA) 2024-07-03 EP disclosed
WO-2023023853-A1 TRANSCRIPTION FACTOR BRN2 INHIBITORY COMPOUNDS FOR USE AS THERAPEUTICS THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2023-03-02 WO disclosed
CN-112105654-A Curable resin mixture, curable resin composition, and cured product thereof 日本化药株式会社 2020-12-18 CN disclosed
WO-2020252205-A1 INHIBITORS OF INTEGRATED STRESS RESPONSE PATHWAY Praxis Biotech LLC (US) 2020-12-17 WO disclosed
WO-2020031935-A1 CURABLE RESIN MIXTURE, CURABLE RESIN COMPOSITION, AND CURED PRODUCT 日本化薬株式会社 2020-02-13 WO disclosed
CN-208980610-U 5- chlorine indone process units 宿迁市科莱博生物化学有限公司 2019-06-14 CN disclosed
US-9573939-B2 Substituted benzofuran compounds and methods of use thereof for the treatment of viral diseases MERCK SHARP & DOHME CORP. (US) 2017-02-21 US disclosed
US-9540400-B2 Compounds as diacylglycerol acyltransferase inhibitors GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2017-01-10 US disclosed
WO-2005058836-A1 INSECTICIDAL SPIROINDANE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2005-06-30 WO disclosed
EP-1492749-A1 PREPARATION OF SUBSTITUTED INDENES Basell Polyolefine GmbH (DE) 2005-01-05 EP disclosed
WO-2003084904-A1 PREPARATION OF SUBSTITUTED INDENES BASELL POLYOLEFINE GMBH (DE) 2003-10-16 WO disclosed
US-6087292-A Metallocene catalysts comprising indenyl ligands substituted with electronegative groups TANGOR GMBH (DE) 2000-07-11 US disclosed
US-5763542-A Process for the preparation of an olefin polymer using specific metallocenes TARGOR GMBH (DE) 1998-06-09 US disclosed
EP-0505972-B1 Process for producing styrenic copolymer IDEMITSU KOSAN CO (JP) 1997-06-11 EP disclosed
US-5504232-A Process for the preparation of an olefin polymer using specific metallocenes HOECHST AKTIENGESELLSCHAFT (DE) 1996-04-02 US disclosed
EP-0505972-A2 Process for producing styrenic copolymer IDEMITSU KOSAN COMPANY LIMITED (JP) 1992-09-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060052620-A1 Preparation of substituted indenes INTS9, CYP1A2, INF2 HTR2C 3399/4885HTR2A 3428/4885HTR2B 2637/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.