SCHEMBL17870698

SCHEMBL17870698

CN(C)CCn1c(=O)[nH]cc(Br)c1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.40
PDE4B Q07343 2/20 0.40
PDE4C Q08493 2/20 0.40
PDE4D Q08499 2/20 0.40
MPO P05164 3/20 0.38
HAVCR2 Q8TDQ0 1/20 0.38
TOP2A P11388 1/20 0.37
DAO P14920 1/20 0.37
KDM4E B2RXH2 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PLK1 P53350 1/20 0.33
TDP1 Q9NUW8 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
POLB P06746 1/20 0.33
CSNK2A1 P68400 1/20 0.32
WEE1 P30291 1/20 0.32
DRD2 P14416 1/20 0.32
HTR6 P50406 1/20 0.32
NR3C1 P04150 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15229791 0.72 PDE4A (0.39) PDE4APDE4BPDE4CPDE4DMPO
SCHEMBL16652006 0.70 ADORA2A (0.36) ALDH1A1CSNK2A1
SCHEMBL9725356 0.70 CCR4 (0.43) MPOHAVCR2DAOSMN1; SMN2TDP1
Hydrochloric Acid SCHEMBL9725475 0.69 CCR4 (0.42) MPOHAVCR2DAOSMN1; SMN2ALDH1A1
SCHEMBL7615724 0.69 TSHR (0.35) SMN1; SMN2ALDH1A1
SCHEMBL9725374 0.68 DAO (0.36) PDE4APDE4BPDE4CPDE4DMPO
SCHEMBL9725387 0.68 DAO (0.36) PDE4APDE4BPDE4CPDE4DMPO
SCHEMBL29099240 0.68 DAO (0.47) PDE4APDE4BPDE4CPDE4DMPO
Hydrochloric Acid SCHEMBL9725534 0.67 DAO (0.35) PDE4APDE4BPDE4CPDE4DMPO
Hydrochloric Acid SCHEMBL9725460 0.67 DAO (0.35) PDE4APDE4BPDE4CPDE4DMPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3237403-A1 NOVEL HETEROCYCLIC COMPOUNDS AND THE USE THEREOF IN MEDICINE AND IN COSMETICS Galderma Research & Development (FR) 2017-11-01 EP disclosed
WO-2016102882-A1 NOVEL HETEROCYCLIC COMPOUNDS AND THE USE THEREOF IN MEDICINE AND IN COSMETICS GALDERMA RESEARCH & DEVELOPMENT (FR) 2016-06-30 WO disclosed