SCHEMBL17874

SCHEMBL17874

O=C(O)CC(S[Au])C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.43
CPB1 P15086 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
SLC22A6 Q4U2R8 1/20 0.39
ALDH1A1 P00352 3/20 0.39
POLB P06746 3/20 0.39
CYP2C19 P33261 2/20 0.39
CYP2C9 P11712 1/20 0.39
KDM4E B2RXH2 2/20 0.38
APOBEC3G Q9HC16 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
FOLH1 Q04609 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAPT P10636 1/20 0.34
BHMT Q93088 1/20 0.34
GABRR1 P24046 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5188914 0.97 TDP1 (0.42) TDP1CPB1SMN1; SMN2SLC22A6ALDH1A1
SCHEMBL7780055 0.80 TDP1 (0.40) TDP1CPB1SMN1; SMN2SLC22A6ALDH1A1
SCHEMBL8948260 0.79 TDP1 (0.50) TDP1CPB1SMN1; SMN2SLC22A6ALDH1A1
SCHEMBL17372820 0.78 CA2 (0.36) TDP1CPB1SMN1; SMN2SLC22A6NPSR1
SCHEMBL630577 0.78 TDP1 (0.48) TDP1CPB1SMN1; SMN2SLC22A6ALDH1A1
SCHEMBL10729283 0.78 TDP1 (0.48) TDP1CPB1SMN1; SMN2SLC22A6ALDH1A1
SCHEMBL7720554 0.76 TDP1 (0.46) TDP1CPB1SMN1; SMN2SLC22A6ALDH1A1
Hydrogen Sulfide SCHEMBL11546403 0.76 TDP1 (0.46) TDP1CPB1SMN1; SMN2SLC22A6ALDH1A1
SCHEMBL233153 0.75 TDP1 (0.40) TDP1CPB1SMN1; SMN2SLC22A6ALDH1A1
SCHEMBL630522 0.75 SMN1; SMN2 (0.44) TDP1CPB1SMN1; SMN2SLC22A6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2553 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3829569-B1 SPINOSYN FORMULATIONS FOR USE IN THE TREATMENT OF DEMODEX-INDUCED OCULAR CONDITIONS APERTA BIOSCIENCES LLC (US) 2025-09-03 EP claimed
US-12337065-B2 Compositions for treating viral infections and methods for same ACCESS TO ADVANCED HEALTH INSTITUTE (US) 2025-06-24 US claimed
US-12297294-B2 Cortistatin analogues for the treatment of inflammatory and/or immune diseases BCN PEPTIDES, S.A. (ES) 2025-05-13 US claimed
EP-4543898-A1 PYRIMIDINE NUCLEOSIDE TREATMENTS The Children's Medical Center Corporation (US) 2025-04-30 EP claimed
EP-4365189-B1 PREVENTION OF DISULFIDE BOND REDUCTION DURING RECOMBINANT PRODUCTION OF POLYPEPTIDES HOFFMANN LA ROCHE (CH) 2025-02-19 EP claimed
EP-4365189-A2 PREVENTION OF DISULFIDE BOND REDUCTION DURING RECOMBINANT PRODUCTION OF POLYPEPTIDES GENENTECH, INC. (US) 2024-05-08 EP claimed
EP-4335863-A2 PREVENTION OF DISULFIDE BOND REDUCTION DURING RECOMBINANT PRODUCTION OF POLYPEPTIDES Genentech, Inc. (US) 2024-03-13 EP claimed
US-20240075047-A1 aPKC INHIBITORS AND METHODS OF TREATING A NEURODEGENERATIVE DISEASE OR DISORDER THE UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS 2024-03-07 US claimed
EP-4245766-A9 PREVENTION OF DISULFIDE BOND REDUCTION DURING RECOMBINANT PRODUCTION OF POLYPEPTIDES Genentech, Inc. (US) 2024-01-24 EP claimed
US-11865125-B2 APKC inhibitors and methods of treating a neurodegenerative disease or disorder UNIVERSITY OF SOUTH FLORIDA (US) 2024-01-09 US claimed
WO-2005123193-A2 TREATMENTS COMPRISING STRONTIUM FOR RHEUMATIC AND ARTHRITIC DISEASES AND PAIN OSTEOLOGIX A/S (DK) 2005-12-29 WO claimed
WO-2005108339-A2 HIGH YIELD AND RAPID SYNTHESES METHODS FOR PRODUCING METALLO-ORGANIC SALTS OSTEOLOGIX A/S (DK) 2005-11-17 WO claimed
US-6914128-B1 Comprises immunoglobulin for treatment and prevention of inflammatory and autoimmune diseases ABBOTT GMBH & CO. KG (DE) 2005-07-05 US claimed
WO-2004045505-A2 EXTRACT OF STEPHANIAE SINICA DIELS AND METHODS OF USING THE SAME WONG KIN-PING (US) 2004-06-03 WO claimed
WO-2004043346-A2 COMPOSITIONS CONTAINING AN ACTIVE FRACTION ISOLATED FROM LYCIUM BARBARUM AND METHODS OF USING THE SAME WONG KIN-PING (US) 2004-05-27 WO claimed
WO-2001021190-A9 TREATMENT FOR NARCOLEPSY UNIV CALIFORNIA (US) 2002-07-11 WO claimed
WO-2001021190-A1 TREATMENT FOR NARCOLEPSY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2001-03-29 WO claimed
US-6204245-B1 Treatment of narcolepsy with immunosuppressants THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2001-03-20 US claimed
EP-0427843-B1 SPECIFIC INHIBITOR FOR RETROVIRUS REVERSE TRANSCRIPTASE, AND ITS APPLICATION AS A MEDICAMENT BLOUGH HERBERT A (US) 1995-03-08 EP claimed
US-4265823-A GOLD COMPOUNDS POSSESSING ANTIINFLAMMATORY PROPERTIES Kosinski, Robert E. (US) 1981-05-05 US claimed