SCHEMBL17895130

SCHEMBL17895130

COc1ccc(CNCCc2cc(C)c(C(=O)O)cn2)c(OC)c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.52
MAPT P10636 2/20 0.51
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.49
APLNR P35414 1/20 0.49
TAS1R3 Q7RTX0 2/20 0.48
TAS1R1 Q7RTX1 2/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
ALDH1A1 P00352 1/20 0.47
TSHR P16473 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
CD274 Q9NZQ7 2/20 0.43
P4HTM Q9NXG6 1/20 0.43
PDCD1 Q15116 1/20 0.43
DPP7 Q9UHL4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15878428 0.81 TAS1R3 (0.52) KDM4CMAPTHTR2AHTR2CAPLNR
SCHEMBL22556655 0.75 APLNR (0.65) HTR2AHTR2CAPLNRTAS1R3TAS1R1
SCHEMBL16343541 0.73 KDM4C (0.64) KDM4CMAPTAPLNRTAS1R3TAS1R1
SCHEMBL1493653 0.73 MAPT (0.59) KDM4CMAPTMEN1KMT2AALDH1A1
SCHEMBL3200678 0.73 APLNR (0.67) KDM4CHTR2AHTR2CAPLNRTAS1R3
SCHEMBL20565881 0.73 APLNR (0.61) HTR2AHTR2CAPLNRTAS1R3TAS1R1
SCHEMBL22657816 0.73 APLNR (0.66) KDM4CMAPTAPLNRTAS1R3TAS1R1
SCHEMBL29444046 0.73 APLNR (0.66) KDM4CMAPTAPLNRTAS1R3TAS1R1
SCHEMBL7768853 0.72 APLNR (0.86) HTR2AHTR2CAPLNRMEN1KMT2A
SCHEMBL701192 0.72 TAS1R3 (0.86) MAPTAPLNRTAS1R3TAS1R1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016106628-A1 BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-07-07 WO disclosed