SCHEMBL17896702

SCHEMBL17896702

Cc1cncc(-c2nc3cc(F)cc(F)c3n2C)c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 11/20 0.41
CYP11B1 P15538 10/20 0.41
PTGS2 P35354 2/20 0.37
CYP19A1 P11511 2/20 0.36
ADRA2B P18089 1/20 0.36
TDO2 P48775 1/20 0.35
PIK3CA P42336 1/20 0.33
PDE2A O00408 1/20 0.33
PDE10A Q9Y233 1/20 0.33
DHODH Q02127 1/20 0.33
CYP2A6 P11509 2/20 0.33
MET P08581 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896600 0.90 CYP11B2 (0.45) CYP11B2CYP11B1CYP19A1ADRA2B
SCHEMBL17896699 0.86 PTGS2 (0.39) CYP11B2CYP11B1PTGS2CYP19A1ADRA2B
SCHEMBL17896703 0.84 CYP11B1 (0.50) CYP11B2CYP11B1PTGS2PDE2APDE10A
SCHEMBL17896704 0.83 CYP11B2 (0.49) CYP11B2CYP11B1
SCHEMBL17896700 0.81 CYP11B2 (0.62) CYP11B2CYP11B1
SCHEMBL10175459 0.79 CYP11B2 (0.56) CYP11B2CYP11B1PTGS2CYP19A1ADRA2B
SCHEMBL10175431 0.77 CYP11B1 (0.42) CYP11B2CYP11B1PTGS2CYP19A1ADRA2B
SCHEMBL460559 0.77 CYP11B2 (0.46) CYP11B2CYP11B1CYP19A1PDE2APDE10A
SCHEMBL17883792 0.77 CYP11B2 (0.58) CYP11B2CYP11B1CYP19A1ADRA2B
SCHEMBL10176203 0.74 CYP11B2 (0.69) CYP11B2CYP11B1CYP19A1ADRA2BTDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed