SCHEMBL17896704

SCHEMBL17896704

Cn1c(-c2cncc(C#N)c2)nc2cc(F)cc(F)c21

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 8/20 0.49
CYP11B1 P15538 5/20 0.49
SSTR5 P35346 1/20 0.40
NPY5R Q15761 1/20 0.36
TLR7 Q9NYK1 7/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896600 0.84 CYP11B2 (0.45) CYP11B2CYP11B1TLR7CHRNB2CHRNB4
SCHEMBL17896702 0.83 CYP11B2 (0.41) CYP11B2CYP11B1
SCHEMBL10175455 0.81 CYP11B2 (0.51) CYP11B2CYP11B1SSTR5NPY5RTLR7
SCHEMBL17896699 0.81 PTGS2 (0.39) CYP11B2CYP11B1TLR7
SCHEMBL10175146 0.80 CYP11B2 (0.67) CYP11B2CYP11B1
SCHEMBL17896703 0.79 CYP11B1 (0.50) CYP11B2CYP11B1
SCHEMBL17896700 0.75 CYP11B2 (0.62) CYP11B2CYP11B1
SCHEMBL17896609 0.73 CYP11B2 (0.48) CYP11B2CYP11B1
SCHEMBL460559 0.72 CYP11B2 (0.46) CYP11B2CYP11B1SSTR5
SCHEMBL462661 0.72 CYP11B2 (0.46) CYP11B2CYP11B1SSTR5TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed