SCHEMBL17896756

SCHEMBL17896756

COc1cncc(-c2nc3cc(NS(C)(=O)=O)ccc3n2C)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.45
ALOX5AP P20292 1/20 0.45
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
ALDH1A1 P00352 3/20 0.43
TP53 P04637 2/20 0.43
LMNA P02545 2/20 0.43
POLB P06746 1/20 0.43
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
KIT P10721 1/20 0.42
BRPF1 P55201 1/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
KDM4E B2RXH2 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10175614 0.84 SMN1; SMN2 (0.46) CA12CA1CA2CA9SMN1; SMN2
SCHEMBL17896755 0.84 SMN1; SMN2 (0.44) CA12CA1CA2CA9SMN1; SMN2
SCHEMBL17896649 0.83 PTGS2 (0.58) PTGS2ALOX5APCA12CA1CA2
SCHEMBL17896760 0.81 CYP11B1 (0.52) PTGS2ALOX5APCA12CA1CA2
SCHEMBL460529 0.81 NAMPT (0.53) PTGS2ALOX5APSMN1; SMN2ALDH1A1LMNA
SCHEMBL17896621 0.78 SMN1; SMN2 (0.49) PTGS2ALOX5APCA12CA1CA2
SCHEMBL17896664 0.78 ALOX5AP (0.54) PTGS2ALOX5APCA12CA1CA2
SCHEMBL10175433 0.78 CYP11B1 (0.53) PTGS2ALOX5APCA12CA1CA2
SCHEMBL17896642 0.75 ALOX5AP (0.46) PTGS2ALOX5APCA12CA1CA2
SCHEMBL17896627 0.75 PTGS2 (0.51) PTGS2ALOX5APCYP11B1CYP11B2KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed