SCHEMBL17896642

SCHEMBL17896642

COc1cncc(-c2nc3cc(C#N)ccc3n2C)c1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 2/20 0.46
CYP11B2 P19099 7/20 0.45
CYP11B1 P15538 6/20 0.45
PDE2A O00408 1/20 0.42
PDE10A Q9Y233 1/20 0.42
KDM1A O60341 1/20 0.41
PTGER4 P35408 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
SCN9A Q15858 1/20 0.39
PTGS2 P35354 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896611 0.91 CYP11B2 (0.50) ALOX5APCYP11B2CYP11B1PDE2APDE10A
SCHEMBL10175348 0.85 CYP11B2 (0.48) CYP11B2CYP11B1PTGER4CA12CA1
SCHEMBL17896760 0.85 CYP11B1 (0.52) ALOX5APCYP11B2CYP11B1PDE2APDE10A
SCHEMBL17896643 0.84 CYP11B2 (0.66) CYP11B2CYP11B1
SCHEMBL10175342 0.83 CYP11B2 (0.46) CYP11B2CYP11B1PTGER4PTGS2CA12
SCHEMBL17896641 0.83 CYP11B2 (0.47) CYP11B2CYP11B1PTGER4
SCHEMBL17896664 0.81 ALOX5AP (0.54) ALOX5APCYP11B2CYP11B1PDE2APDE10A
SCHEMBL10175433 0.81 CYP11B1 (0.53) ALOX5APCYP11B2CYP11B1PDE2APDE10A
SCHEMBL17896621 0.81 SMN1; SMN2 (0.49) ALOX5APCYP11B2CYP11B1PDE2APDE10A
SCHEMBL17883795 0.80 CYP11B2 (0.47) CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed