SCHEMBL17898768

SCHEMBL17898768

COc1ccnc(C(=O)N[C@H]2CCCC[C@H](Cc3ccccc3)[C@@H](OCC(C)C)[C@H](C)OC2=O)c1O

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.33
TAS1R1 Q7RTX1 2/20 0.33
ABCB1 P08183 1/20 0.31
CTSK P43235 2/20 0.31
RIPK1 Q13546 3/20 0.30
ADORA2A P29274 1/20 0.30
HCRTR1 O43613 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16605191 0.98 TAS1R3 (0.33) TAS1R3TAS1R1ABCB1CTSKRIPK1
SCHEMBL16605203 0.92 HPGDS (0.32)
SCHEMBL16605214 0.92
SCHEMBL16605185 0.91 HCRTR1 (0.33) TAS1R3TAS1R1RIPK1HCRTR1
SCHEMBL17898782 0.91 RIPK1 (0.33) RIPK1
SCHEMBL17898764 0.91 RIPK1 (0.33) CTSKRIPK1
SCHEMBL16605196 0.90 TAS1R3 (0.35) TAS1R3TAS1R1RIPK1ADORA2AHCRTR1
SCHEMBL16605197 0.90 TAS1R3 (0.35) TAS1R3TAS1R1RIPK1ADORA2AHCRTR1
SCHEMBL15530250 0.90 ABCB1 (0.31) ABCB1RIPK1
SCHEMBL15366272 0.90 ABCB1 (0.31) ABCB1RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016109291-A1 USE OF MACROCYCLIC PICOLINAMIDES AS FUNGICIDES DOW AGROSCIENCES LLC (US) 2016-07-07 WO disclosed
WO-2016109290-A1 MACROCYCLIC PICOLINAMIDE COMPOUNDS WITH FUNGICIDAL ACTIVITY DOW AGROSCIENCES LLC (US) 2016-07-07 WO disclosed