SCHEMBL17898781

SCHEMBL17898781

CC[C@H]1CCOC[C@H](NC(=O)c2nccc(OC)c2OC(C)=O)C(=O)O[C@@H](C)[C@@H]1OC(=O)c1ccccc1

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.32
RIPK1 Q13546 1/20 0.31
PTPN1 P18031 1/20 0.31
OPRM1 P35372 1/20 0.30
OPRD1 P41143 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17899036 0.90 ROCK1 (0.31) ROCK1RIPK1PTPN1
SCHEMBL19089232 0.88 RIPK1 (0.32) ROCK1RIPK1
SCHEMBL19088922 0.85 RIPK1 (0.35) ROCK1RIPK1
SCHEMBL17898884 0.83 ROCK1 (0.31) ROCK1RIPK1
SCHEMBL17898759 0.82
SCHEMBL19089231 0.82 PDE4D (0.34)
SCHEMBL19091284 0.82 RIPK1 (0.33) RIPK1
SCHEMBL17899016 0.82 IGF1R (0.32) RIPK1
SCHEMBL17898822 0.82 RIPK1 (0.32) RIPK1
SCHEMBL19091513 0.81 MERTK (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016109291-A1 USE OF MACROCYCLIC PICOLINAMIDES AS FUNGICIDES DOW AGROSCIENCES LLC (US) 2016-07-07 WO disclosed
WO-2016109290-A1 MACROCYCLIC PICOLINAMIDE COMPOUNDS WITH FUNGICIDAL ACTIVITY DOW AGROSCIENCES LLC (US) 2016-07-07 WO disclosed