SCHEMBL17899036

SCHEMBL17899036

CC[C@H]1CCOC[C@H](NC(=O)c2nccc(OC)c2O)C(=O)O[C@@H](C)[C@@H]1OC(=O)c1ccccc1

nearest known ligand 0.31

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.31
HPGDS O60760 1/20 0.31
RIPK1 Q13546 1/20 0.31
DRD2 P14416 1/20 0.31
TAS1R3 Q7RTX0 2/20 0.30
TAS1R1 Q7RTX1 2/20 0.30
PDCD1 Q15116 2/20 0.30
CD274 Q9NZQ7 2/20 0.30
PTPN1 P18031 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17898781 0.90 ROCK1 (0.32) ROCK1RIPK1PTPN1
SCHEMBL17898894 0.90 HPGDS (0.32) ROCK1HPGDSRIPK1TAS1R3TAS1R1
SCHEMBL17899031 0.89 HPGDS (0.31) HPGDS
SCHEMBL19088927 0.88 TAS1R3 (0.33) ROCK1HPGDSRIPK1TAS1R3TAS1R1
SCHEMBL15373323 0.87 ABCB1 (0.31) RIPK1PTPN1
SCHEMBL17898885 0.87 BCHE (0.33) HPGDS
SCHEMBL17898692 0.85 HPGDS (0.30) HPGDS
SCHEMBL19088921 0.84 RIPK1 (0.36) RIPK1TAS1R3TAS1R1
SCHEMBL15373823 0.83 BCHE (0.34) PTPN1
SCHEMBL19088924 0.83 PDE4D (0.36) RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016109291-A1 USE OF MACROCYCLIC PICOLINAMIDES AS FUNGICIDES DOW AGROSCIENCES LLC (US) 2016-07-07 WO disclosed
WO-2016109290-A1 MACROCYCLIC PICOLINAMIDE COMPOUNDS WITH FUNGICIDAL ACTIVITY DOW AGROSCIENCES LLC (US) 2016-07-07 WO disclosed