SCHEMBL17898786

SCHEMBL17898786

C(#Cc1ccc2ccc3ccc(C#Cc4cccnc4)cc3c2c1)c1cccnc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 6/20 0.50
CYP2A6 P11509 4/20 0.50
AAK1 Q2M2I8 1/20 0.50
CYP2D6 P10635 3/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2C9 P11712 3/20 0.49
CYP2B6 P20813 3/20 0.49
CYP2C19 P33261 3/20 0.49
CYP2E1 P05181 2/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2C8 P10632 1/20 0.47
KCNH2 Q12809 1/20 0.47
PIK3CA P42336 2/20 0.46
PDK1 Q15118 1/20 0.46
CHRNB2 P17787 2/20 0.46
CHRNA4 P43681 2/20 0.46
FFAR1 O14842 1/20 0.45
MTOR P42345 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13907278 0.82 CYP2A6 (0.62) GRM5CYP2A6CYP2D6CYP1A2CYP2C9
SCHEMBL3796332 0.82 CYP2A6 (0.67) GRM5CYP2A6CYP2D6CYP1A2CYP2C9
SCHEMBL1476884 0.76 CYP2A6 (0.49) GRM5CYP2A6CYP2D6CYP1A2CYP2C9
SCHEMBL401836 0.76 GRM5 (0.64) GRM5CYP2A6CYP2D6CYP1A2CYP2C9
SCHEMBL31673222 0.76 GRM5 (0.64) GRM5CYP2A6CYP2D6CYP1A2CYP2C9
SCHEMBL1477031 0.74 GRM5 (0.50) GRM5CYP2A6CYP2D6CYP1A2CYP2C9
SCHEMBL2806708 0.74 MEN1 (0.55) GRM5CYP2A6CYP2D6CYP1A2CYP2C9
SCHEMBL31673182 0.74 GRM5 (0.71) GRM5CYP2A6CYP2D6CYP1A2CYP2C9
SCHEMBL2806200 0.74 CYP2A6 (0.50) GRM5CYP2A6CYP2D6CYP1A2CYP2C9
SCHEMBL1477185 0.74 GRM5 (0.50) GRM5CYP2A6CYP2D6CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016108489-A1 NOVEL RUTHENIUM COMPOUND, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING CANCER, CONTAINING SAME AS ACTIVE INGREDIENT 울산대학교 산학협력단 2016-07-07 WO disclosed