SCHEMBL17907922

SCHEMBL17907922

CC(C)(C)OC(=O)C1C(=O)CCc2cc3cc(OC(F)(F)F)ccc3n21

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 2/20 0.38
KCNQ2 O43526 2/20 0.38
IDH1 O75874 12/20 0.37
LIPE Q05469 1/20 0.35
GPR119 Q8TDV5 1/20 0.34
PIM1 P11309 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17907981 0.88 KDM4E (0.39)
SCHEMBL17907954 0.84 NR1H2 (0.36)
SCHEMBL17907924 0.83 NR1H2 (0.35) GPR119
SCHEMBL17907949 0.82 GABRA1 (0.35)
SCHEMBL3542987 0.81 NOTUM (0.40)
SCHEMBL17907968 0.78 HDAC1 (0.34) GPR119
SCHEMBL17907950 0.78 MAPK1 (0.33)
SCHEMBL13279458 0.76 CCR9 (0.34)
SCHEMBL1770176 0.70 KDM4E (0.34) GPR119
SCHEMBL17907935 0.67 MAOA (0.36) PIM1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697223-B1 7-(HETEROARYL-AMINO)-6,7,8,9-TETRAHYDROPYRIDO[1,2-A]INDOL ACETIC ACID DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2016-07-13 EP disclosed