SCHEMBL17907935

SCHEMBL17907935

O=C1CCc2cc3cc(OC(F)(F)F)ccc3n2C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.36
PIM1 P11309 1/20 0.35
CES1 P23141 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
GPR3 P46089 1/20 0.33
F2RL3 Q96RI0 1/20 0.32
CHRM5 P08912 2/20 0.32
KDM4E B2RXH2 2/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
POLB P06746 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CYP2D6 P10635 1/20 0.32
KCNN4 O15554 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GRIN2B Q13224 1/20 0.32
S1PR1 P21453 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17907920 0.82 HTR2A (0.51) HTR2AHTR2CKDM4EGAAKMT2A
SCHEMBL17907947 0.70 ALDH1A1 (0.38) KMT2AL3MBTL1
SCHEMBL3155248 0.70 HTR2C (0.69) MAOAPIM1HTR2AHTR2CS1PR1
SCHEMBL17907922 0.67 KCNQ3 (0.38) PIM1CYP2D6
SCHEMBL6713758 0.66 HTR2C (0.51) PIM1HTR2AHTR2C
SCHEMBL17907965 0.65 HTR2A (0.48) HTR2AHTR2CKMT2A
SCHEMBL17310928 0.65 F2RL3 (0.43) PIM1GPR3F2RL3KDM4EKMT2A
SCHEMBL8060053 0.63 CYP2A6 (0.44) CES1GPR3CHRM5KDM4ECRHBP
SCHEMBL10253811 0.61 KDM4E (0.69) PIM1F2RL3KDM4EGAAKMT2A
SCHEMBL2439728 0.60 NOTUM (0.50) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697223-B1 7-(HETEROARYL-AMINO)-6,7,8,9-TETRAHYDROPYRIDO[1,2-A]INDOL ACETIC ACID DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2016-07-13 EP disclosed