SCHEMBL17907933

SCHEMBL17907933

CC(C)(C)OC(=O)Cn1c(/C=C/C(=O)O)cc2cc(OC(F)(F)F)ccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 1/20 0.38
KCNQ2 O43526 1/20 0.38
CACNA1B Q00975 1/20 0.38
NTRK1 P04629 3/20 0.38
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37
THRB P10828 1/20 0.37
IDH1 O75874 3/20 0.37
CNR1 P21554 1/20 0.36
KMT2A Q03164 1/20 0.36
APP P05067 1/20 0.36
AKR1C3 P42330 2/20 0.36
PIM1 P11309 1/20 0.36
IP6K1 Q92551 1/20 0.35
IP6K3 Q96PC2 1/20 0.35
IP6K2 Q9UHH9 1/20 0.35
ESR1 P03372 1/20 0.35
ELANE P08246 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17907934 1.00 KCNQ3 (0.38) KCNQ3KCNQ2CACNA1BNTRK1ALDH1A1
SCHEMBL17907985 0.89 KDM4E (0.41) CACNA1BALDH1A1KDM4ETHRB
SCHEMBL17907984 0.89 KDM4E (0.41) CACNA1BALDH1A1KDM4ETHRB
SCHEMBL17907927 0.86 CACNA1B (0.44) CACNA1BALDH1A1KDM4EKMT2A
SCHEMBL17907928 0.86 CACNA1B (0.44) CACNA1BALDH1A1KDM4EKMT2A
SCHEMBL17907996 0.86 CACNA1B (0.40) CACNA1BNTRK1ALDH1A1KDM4EESR1
SCHEMBL17907997 0.86 CACNA1B (0.40) CACNA1BNTRK1ALDH1A1KDM4EESR1
SCHEMBL17907951 0.85 TDP1 (0.41) CACNA1BALDH1A1KDM4ETHRB
SCHEMBL17907953 0.85 TDP1 (0.41) CACNA1BALDH1A1KDM4ETHRB
SCHEMBL3553079 0.83 KDM4E (0.46) CACNA1BALDH1A1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697223-B1 7-(HETEROARYL-AMINO)-6,7,8,9-TETRAHYDROPYRIDO[1,2-A]INDOL ACETIC ACID DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2016-07-13 EP disclosed