SCHEMBL17928601

SCHEMBL17928601

CCC1COc2cnc3ccc(OC)cc3c2C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 4/20 0.47
CYP1A2 P05177 3/20 0.42
HSD17B10 Q99714 3/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C19 P33261 2/20 0.42
TSHR P16473 2/20 0.42
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.40
MAPT P10636 2/20 0.40
CYP2D6 P10635 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.39
CLK1 P49759 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KCNH2 Q12809 4/20 0.38
ABCB1 P08183 1/20 0.38
ABCC1 P33527 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
PDE5A O76074 1/20 0.38
NCF1 P14598 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12692897 0.91 PDE5A (0.39) MTNR1ACYP1A2HSD17B10CYP3A4CYP2C19
SCHEMBL14250228 0.89 MTNR1A (0.46) MTNR1ACYP1A2HSD17B10CYP3A4CYP2C19
SCHEMBL15960993 0.89 MTNR1A (0.44) MTNR1ACYP1A2HSD17B10CYP3A4CYP2C19
SCHEMBL12692892 0.89 MTNR1A (0.37) MTNR1ACYP1A2HSD17B10CYP3A4CYP2C19
SCHEMBL14314428 0.88 MTNR1A (0.45) MTNR1ACYP1A2HSD17B10CYP3A4CYP2C19
SCHEMBL12692905 0.88 MTNR1A (0.36) MTNR1ACYP1A2HSD17B10CYP3A4CYP2C19
SCHEMBL12692893 0.87 MTNR1A (0.38) MTNR1ACYP1A2HSD17B10CYP3A4CYP2C19
SCHEMBL12692915 0.85 MTNR1A (0.37) MTNR1ACYP1A2HSD17B10CYP3A4CYP2C19
SCHEMBL12630208 0.84 ALDH1A1 (0.43) MTNR1ACYP1A2HSD17B10CYP3A4CYP2C19
SCHEMBL15305097 0.84 ALDH1A1 (0.43) MTNR1ACYP1A2HSD17B10CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2721034-B1 N-HETEROTRICYCLIC ANTIBIOTICS BASILEA PHARMACEUTICA AG (CH) 2016-07-20 EP disclosed