SCHEMBL17957134

SCHEMBL17957134

Cc1c([N+](=O)[O-])ccc2cc(C(=O)O)n(C)c12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.45
MCL1 Q07820 2/20 0.43
CASP6 P55212 1/20 0.41
CCR2 P41597 1/20 0.41
ALDH1A1 P00352 4/20 0.40
KDM4E B2RXH2 3/20 0.40
HPGD P15428 3/20 0.40
HSD17B10 Q99714 3/20 0.40
TDP1 Q9NUW8 2/20 0.40
GPR35 Q9HC97 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
DTYMK P23919 1/20 0.38
CYP3A4 P08684 1/20 0.38
POLB P06746 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
GAA P10253 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
HCAR3 P49019 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13684476 0.82 NOD2 (0.44) ALDH1A1KDM4EHPGDL3MBTL1SMN1; SMN2
SCHEMBL3255649 0.82 CCR2 (0.55) TSHRMCL1CCR2ALDH1A1KDM4E
SCHEMBL26581762 0.80 MCL1 (0.49) MCL1CCR2ALDH1A1KDM4EHPGD
SCHEMBL28461196 0.74 CCR2 (0.45) TSHRCASP6CCR2ALDH1A1KDM4E
SCHEMBL3021221 0.72 ALDH1A1 (0.41) MCL1CCR2ALDH1A1KDM4EHPGD
SCHEMBL8985891 0.72 MCL1 (0.55) MCL1CCR2ALDH1A1KDM4EHPGD
SCHEMBL10233030 0.70 MCL1 (0.57) TSHRMCL1CCR2ALDH1A1KDM4E
SCHEMBL26683715 0.70 TSHR (0.44) TSHRCASP6ALDH1A1TDP1L3MBTL1
SCHEMBL31060526 0.69 MCL1 (0.47) MCL1CCR2ALDH1A1KDM4EHPGD
SCHEMBL23809519 0.69 MCL1 (0.44) MCL1CCR2ALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2522657-B1 INDOLE DERIVATIVE TAKEDA PHARMACEUTICAL (JP) 2016-08-03 EP disclosed