SCHEMBL1796209

SCHEMBL1796209

CON=CNC(=O)c1ccc(C=NO)cc1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
HPGD P15428 2/20 0.38
MAPT P10636 6/20 0.37
KMT2A Q03164 4/20 0.37
GFER P55789 2/20 0.37
SRC P12931 1/20 0.37
NPC1 O15118 4/20 0.36
RAB9A P51151 4/20 0.36
POLB P06746 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TP53 P04637 1/20 0.36
PAX8 Q06710 1/20 0.36
KLF5 Q13887 1/20 0.36
HIF1A Q16665 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KDM4E B2RXH2 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1800343 0.86 ALDH1A1 (0.41) ALDH1A1HPGDMAPTSRCRAB9A
SCHEMBL1796295 0.80 LMNA (0.41) ALDH1A1HPGDMAPTKMT2AGFER
SCHEMBL1800400 0.80 FLT1 (0.44) ALDH1A1HPGDMAPTKMT2ANPC1
SCHEMBL1796296 0.80 LMNA (0.41) ALDH1A1HPGDMAPTKMT2AGFER
SCHEMBL3123464 0.79 NPC1 (0.48) ALDH1A1HPGDMAPTKMT2AGFER
SCHEMBL30008909 0.79 NPC1 (0.48) ALDH1A1HPGDMAPTKMT2AGFER
SCHEMBL3123458 0.79 NPC1 (0.48) ALDH1A1HPGDMAPTKMT2AGFER
SCHEMBL14963072 0.79 NPC1 (0.48) ALDH1A1HPGDMAPTKMT2AGFER
SCHEMBL28897023 0.76 HPGD (0.48) ALDH1A1HPGDMAPTKMT2ANPC1
SCHEMBL27909171 0.76 HPGD (0.48) ALDH1A1HPGDMAPTKMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8987464-B2 Isoxazoline-substituted benzamide compound and pesticide NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2015-03-24 US disclosed
US-20140135496-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2014-05-15 US disclosed
US-8673951-B2 Isoxazoline-substituted benzamide compound and pesticide NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2014-03-18 US disclosed
EP-1932836-B1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND HARMFUL ORGANISM-CONTROLLING AGENT NISSAN CHEMICAL IND LTD (JP) 2013-11-06 EP disclosed
US-20110144334-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2011-06-16 US disclosed
US-7951828-B1 Isoxazoline-substituted benzamide compound and pesticide NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2011-05-31 US disclosed
EP-1932836-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND HARMFUL ORGANISM-CONTROLLING AGENT Nissan Chemical Industries, Ltd. (JP) 2008-06-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110144334-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE OR10J3, OR51E2, ORMDL3 ALDH1A1 475/4885HPGD 3450/4885MAPT 4464/4885
US-20140135496-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE OR10J3, OR51E2, ODC1 ALDH1A1 988/4885HPGD 3906/4885MAPT 3914/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.