SCHEMBL1797222

SCHEMBL1797222

Cc1cc(-c2cccnc2)cc(C(=O)Nc2ccnc(Cl)c2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMARCA2 P51531 3/20 0.49
SMARCA4 P51532 3/20 0.49
PORCN Q9H237 2/20 0.47
IRAK4 Q9NWZ3 1/20 0.47
ABL1 P00519 5/20 0.47
BCR P11274 5/20 0.47
SRC P12931 2/20 0.47
PDGFRB P09619 3/20 0.46
PDGFRA P16234 3/20 0.46
PPARG P37231 1/20 0.45
CYP11B2 P19099 1/20 0.44
CNR1 P21554 1/20 0.44
KDR P35968 1/20 0.44
GRM5 P41594 1/20 0.44
PRKCA P17252 1/20 0.43
PRKCD Q05655 1/20 0.43
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1798177 0.91 GRM5 (0.53) SMARCA2SMARCA4PORCNIRAK4ABL1
SCHEMBL1794228 0.88 SMARCA2 (0.58) SMARCA2SMARCA4GRM5
SCHEMBL1795623 0.87 SMARCA2 (0.49) SMARCA2SMARCA4GRM5CYP1A2CYP3A4
SCHEMBL1794469 0.86 SMARCA2 (0.56) SMARCA2SMARCA4GRM5
SCHEMBL1796453 0.85 SMARCA2 (0.61) SMARCA2SMARCA4PORCNGRM5
SCHEMBL1798156 0.85 CYP1A2 (0.48) SMARCA2SMARCA4GRM5CYP1A2CYP3A4
SCHEMBL1798756 0.83 GRM5 (0.54) SMARCA2SMARCA4GRM5CYP1A2CYP3A4
SCHEMBL1792980 0.82 GRM5 (0.58) SMARCA2SMARCA4PPARGGRM5CYP1A2
SCHEMBL1797503 0.81 SMARCA2 (0.60) SMARCA2SMARCA4PORCNGRM5MEN1
SCHEMBL1794792 0.81 GRM5 (0.50) PPARGGRM5CYP1A2CYP2C9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7951824-B2 4-aryl-pyridine-2-carboxyamide derivatives HOFFMAN-LA ROCHE INC. (US) 2011-05-31 US claimed
US-7951824-B2 4-aryl-pyridine-2-carboxyamide derivatives HOFFMAN-LA ROCHE INC. (US) 2011-05-31 US disclosed