SCHEMBL17992196

SCHEMBL17992196

COc1c2c(nc3c1CCCO3)CCC2

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 14/20 0.58
BCHE P06276 2/20 0.34
APP P05067 1/20 0.34
NPC1 O15118 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MEN1 O00255 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
BPTF Q12830 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
ABCB1 P08183 1/20 0.31
TUBB3 Q13509 1/20 0.31
EHMT2 Q96KQ7 1/20 0.31
HTR2C P28335 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19407334 0.93 ACHE (0.50) ACHEBCHEAPPNPC1KDM4E
SCHEMBL17992288 0.75 ACHE (0.66) ACHEBCHEKDM4EALDH1A1MEN1
SCHEMBL19407545 0.74 ACHE (0.37) ACHE
SCHEMBL17992287 0.74 ACHE (1.00) ACHEBCHEAPPKDM4EALDH1A1
SCHEMBL9584087 0.70 ACHE (1.00) ACHEBCHEAPPKDM4EALDH1A1
SCHEMBL19407388 0.70 ACHE (0.34) ACHE
SCHEMBL2407199 0.64 ACHE (0.37) ACHE
SCHEMBL2407668 0.63 ACHE (0.36) ACHE
SCHEMBL2408242 0.63 ACHE (0.38) ACHEMAPK1
SCHEMBL21938559 0.63 ACHE (0.45) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10696635-B2 Versatile ligand for palladium-catalyzed meta-C—H functionalizations of aromatic substrates THE SCRIPPS RESEARCH INSTITUTE (US) 2020-06-30 US disclosed
US-10611723-B2 Ligand-enabled meta-C-H activation using a transient mediator THE SCRIPPS RESEARCH INSTITUTE (US) 2020-04-07 US disclosed
US-20190119212-A1 A VERSATILE LIGAND FOR PALLADIUM-CATALYZED META-C-H FUNCTIONALIZATIONS THE SCRIPPS RESEARCH INSTITUTE 2019-04-25 US disclosed
WO-2017184589-A1 A VERSATILE LIGAND FOR PALLADIUM-CATALYZED META-C-H FUNCTIONALIZATIONS THE SCRIPPS RESEARCH INSTITUTE (US) 2017-10-26 WO disclosed
WO-2016123361-A1 LIGAND-ENABLED META-C-H ACTIVATION USING A TRANSIENT MEDIATOR THE SCRIPPS RESEARCH INSTITUTE (US) 2016-08-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10611723-B2 Ligand-enabled meta-C-H activation using a transient mediator HRH4, AHR, HRH3 ACHE 659/4885BCHE 402/4885APP 3113/4885
US-20190119212-A1 A VERSATILE LIGAND FOR PALLADIUM-CATALYZED META-C-H FUNCTIONALIZATIONS AHR, PAH, DOHH ACHE 1129/4885BCHE 325/4885APP 2768/4885
US-10696635-B2 Versatile ligand for palladium-catalyzed meta-C—H functionalizations of aromatic substrates PAH, AHR, DDC ACHE 1260/4885BCHE 539/4885APP 2150/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.