SCHEMBL17993499

SCHEMBL17993499

NC(=S)NC(=O)C1(c2ccccc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 3/20 0.53
ALDH1A1 P00352 3/20 0.49
HSD11B1 P28845 2/20 0.47
THRB P10828 1/20 0.47
HDAC1 Q13547 1/20 0.47
HTT P42858 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
AKR1C1 Q04828 1/20 0.46
LMNA P02545 3/20 0.45
NPSR1 Q6W5P4 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ELOVL1 Q9BW60 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
GAA P10253 1/20 0.43
PKM P14618 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2363240 0.82 HDAC4 (0.59) HDAC4ALDH1A1HSD11B1THRBHDAC1
SCHEMBL172001 0.80 HDAC4 (0.50) HDAC4ALDH1A1HSD11B1THRBHDAC1
SCHEMBL1100195 0.78 HDAC4 (0.59) HDAC4ALDH1A1HSD11B1THRBHDAC1
SCHEMBL14019859 0.78 EPHX1 (0.56) HDAC4ALDH1A1HSD11B1THRBHDAC1
SCHEMBL14817498 0.76 SMN1; SMN2 (0.48) HDAC4ALDH1A1HSD11B1THRBHDAC1
SCHEMBL169873 0.76 ALDH1A1 (0.59) HDAC4ALDH1A1HSD11B1THRBHTT
SCHEMBL2722547 0.75 AKR1C1 (0.57) HDAC4HSD11B1THRBHDAC1HTT
SCHEMBL5055163 0.75 AKR1C1 (0.47) HDAC4HSD11B1AKR1C1
SCHEMBL501923 0.75 AKR1C1 (0.57) HDAC4HSD11B1THRBHDAC1HTT
SCHEMBL8572144 0.74 HDAC4 (0.59) HDAC4ALDH1A1HSD11B1THRBHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426108-B1 Processes and intermediates for preparing fused heterocyclic kinase inhibitors METHYLGENE INC (CA) 2016-08-10 EP disclosed