SCHEMBL18015281

SCHEMBL18015281

Brc1cc(-c2ccccc2C2=CC=C(c3ccccn3)CC2)cc(-c2ccccc2-c2ccc(-c3ccccn3)cc2)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.35
CHEK2 O96017 1/20 0.35
PDK2 Q15119 1/20 0.34
EDNRB P24530 1/20 0.34
EDNRA P25101 1/20 0.34
CYP1A2 P05177 2/20 0.33
CYP2D6 P10635 1/20 0.33
CYP19A1 P11511 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KDM4E B2RXH2 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
CCR1 P32246 1/20 0.33
CCR5 P51681 1/20 0.33
CCR8 P51685 1/20 0.33
METAP1 P53582 1/20 0.33
BLM P54132 1/20 0.33
HIF1A Q16665 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18573261 0.87 CCR1 (0.41) GRM5CHEK2PDK2EDNRBEDNRA
SCHEMBL18015564 0.86 KDM4E (0.43) GRM5CHEK2PDK2CYP1A2CYP2D6
SCHEMBL31090826 0.86 KDM4E (0.43) GRM5CHEK2PDK2CYP1A2CYP2D6
SCHEMBL19794394 0.78 KDM4E (0.52) GRM5CHEK2PDK2CYP1A2CYP2D6
SCHEMBL18015184 0.76 ALDH1A1 (0.47) GRM5CHEK2PDK2EDNRBEDNRA
SCHEMBL18015186 0.76 ALDH1A1 (0.47) GRM5CHEK2PDK2EDNRBEDNRA
SCHEMBL25070279 0.75 TGFBR1 (0.49) GRM5PDK2CYP1A2CYP2D6CYP19A1
SCHEMBL17296043 0.75 KDM4E (0.48) GRM5CYP1A2CYP2D6CYP19A1CYP2C9
SCHEMBL9958239 0.73 KDM4E (0.54) GRM5CYP1A2CYP2D6CYP19A1CYP2C9
SCHEMBL21125566 0.73 CYP2A6 (0.46) GRM5CHEK2PDK2CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016124304-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2016-08-11 WO disclosed