SCHEMBL18573261

SCHEMBL18573261

Clc1cc(-c2ccccc2C2=CC=C(c3ccccn3)CC2)cc(-c2ccccc2-c2ccc(-c3ccccn3)cc2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.41
CCR5 P51681 1/20 0.41
CCR8 P51685 1/20 0.41
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
GRM5 P41594 3/20 0.39
TGFBR1 P36897 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CHEK2 O96017 1/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
CASP3 P42574 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18015281 0.87 GRM5 (0.35) CCR1CCR5CCR8PTGS1PTGS2
SCHEMBL18573263 0.86 CCR1 (0.53) CCR1CCR5CCR8ADORA2AADORA1
SCHEMBL19794394 0.78 KDM4E (0.52) CCR1CCR5CCR8GRM5TGFBR1
SCHEMBL21662030 0.76 GRM5 (0.48) CCR1CCR5CCR8GRM5L3MBTL1
SCHEMBL19833337 0.76 CCR1 (0.45) CCR1CCR5CCR8ADORA2AADORA1
SCHEMBL25070279 0.75 TGFBR1 (0.49) CCR1CCR5CCR8GRM5TGFBR1
SCHEMBL19933715 0.75 CCR1 (0.47) CCR1CCR5CCR8ADORA2AADORA1
SCHEMBL23018858 0.75 CCR1 (0.44) CCR1CCR5CCR8ADORA2AADORA1
SCHEMBL20696641 0.74 ABL1 (0.53) CCR1CCR5CCR8PTGS1PTGS2
SCHEMBL16352566 0.73 CCR1 (0.64) CCR1CCR5CCR8ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017032439-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2017-03-02 WO disclosed