SCHEMBL18015693

SCHEMBL18015693

Clc1ccc(-c2ccc(-c3ccccc3-c3cc(-c4ccccc4-c4ccc(-c5ccc(Cl)cc5)nc4)cc(-c4ccccc4-c4ccc(-c5ccc(Cl)cc5)nc4)c3)cn2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
MAP4K4 O95819 1/20 0.45
MAOB P27338 2/20 0.44
KDM1A O60341 1/20 0.44
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HSD17B1 P14061 1/20 0.42
HSD17B2 P37059 1/20 0.42
GRM2 Q14416 1/20 0.42
CTRC Q99895 1/20 0.41
ALOX5 P09917 1/20 0.41
ALDH1A2 O94788 1/20 0.41
ALDH1A3 P47895 1/20 0.41
GAA P10253 1/20 0.40
TGFBR1 P36897 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19933741 0.95 MAP4K4 (0.49) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL18573198 0.90 LDHA (0.45) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL19933709 0.87 TGFBR1 (0.49) MAP4K4HSD17B1HSD17B2CTRCALOX5
SCHEMBL19933578 0.87 LDHA (0.52) HSD17B1HSD17B2LDHA
SCHEMBL18015574 0.87 LDHA (0.52) HSD17B1HSD17B2LDHA
SCHEMBL18015495 0.85 LDHA (0.50) NPC1RAB9ASMN1; SMN2HSD17B1HSD17B2
SCHEMBL19794370 0.85 LDHA (0.50) NPC1RAB9ASMN1; SMN2HSD17B1HSD17B2
SCHEMBL21721920 0.85 LDHA (0.50) HSD17B1HSD17B2LDHA
SCHEMBL19794431 0.85 LDHA (0.50) NPC1RAB9ASMN1; SMN2HSD17B1HSD17B2
SCHEMBL19794427 0.84 CYP2A6 (0.43) NPC1RAB9AMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11024815-B2 Metal complexes MERCK PATENT GMBH (DE) 2021-06-01 US disclosed
EP-3254317-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-07-31 EP disclosed
US-20180026209-A1 Metal Complexes MERCK PATENT GMBH (DE) 2018-01-25 US disclosed
US-20180026209-A1 Metal Complexes MERCK PATENT GMBH (DE) 2018-01-25 US disclosed
WO-2016124304-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2016-08-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11024815-B2 Metal complexes EXOC4, EXOC3, TIMCC NPC1 4039/4885RAB9A 2171/4885SMN1; SMN2 4799/4885
US-20180026209-A1 Metal Complexes AP3M1, AP2M1, SOD1 NPC1 2761/4885RAB9A 1433/4885SMN1; SMN2 4144/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.