SCHEMBL18019207

SCHEMBL18019207

CCC[C@H](NC(=O)OC(C)(C)C)C(=O)NS(=O)(=O)c1cccc(Br)c1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 6/20 0.48
CTSS P25774 4/20 0.48
CTSK P43235 4/20 0.48
CTSB P07858 1/20 0.48
MCL1 Q07820 1/20 0.42
MMP13 P45452 2/20 0.42
AAK1 Q2M2I8 2/20 0.42
CA2 P00918 2/20 0.41
CA1 P00915 1/20 0.41
EGFR P00533 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31650940 0.88 AAK1 (0.57) BCL2CTSSCTSKCTSBMMP13
SCHEMBL19792922 0.88 AAK1 (0.57) BCL2CTSSCTSKCTSBMMP13
SCHEMBL12213922 0.87 BCL2 (0.61) BCL2CTSSCTSKCTSBMCL1
SCHEMBL18019219 0.85 AAK1 (0.59) BCL2CTSSCTSKCTSBMCL1
SCHEMBL18019210 0.82 CA2 (0.57) BCL2CTSSCTSKCTSBAAK1
SCHEMBL1511755 0.81 FLT1 (0.49) CTSSCTSKCTSBCA1EGFR
SCHEMBL31629397 0.81 FLT1 (0.49) CTSSCTSKCTSBCA1EGFR
SCHEMBL19792935 0.78 BCL2 (0.49) BCL2CTSSCTSKCTSBAAK1
SCHEMBL18019121 0.78 CTSK (0.48) BCL2CTSSCTSKCTSBMMP13
SCHEMBL20548447 0.77 BCL2 (0.60) BCL2CTSSCTSKCTSBMCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016129983-A1 NOVEL N-ACYL-ARYLSULFONAMIDE DERIVATIVES AS AMINOACYL-TRNA SYNTHETASE INHIBITORS LATVIAN INSTITUTE OF ORGANIC SYNTHESIS (LV) 2016-08-18 WO disclosed