Tyramine

Tyramine

SCHEMBL1804993

N.NCCc1ccc(O)cc1

nearest known ligand 0.95

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 9/20 0.95
KDM4E B2RXH2 3/20 0.95
ADRA2A P08913 3/20 0.95
SLC6A2 P23975 3/20 0.95
ALDH1A1 P00352 2/20 0.95
HTR1A P08908 2/20 0.95
CYP2C19 P33261 1/20 0.95
HTR3A P46098 1/20 0.95
BACE1 P56817 1/20 0.95
L3MBTL1 Q9Y468 1/20 0.95
TDP1 Q9NUW8 3/20 0.90
BLM P54132 2/20 0.90
KMT2A Q03164 1/20 0.90
ESR1 P03372 2/20 0.65
ESR2 Q92731 2/20 0.65
ABAT P80404 1/20 0.59
CA2 P00918 1/20 0.56
HTR2A P28223 3/20 0.54
CYP2A6 P11509 2/20 0.54
CYP1A2 P05177 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tyramine SCHEMBL134515 0.97 TAAR1 (1.00) TAAR1KDM4EADRA2ASLC6A2ALDH1A1
Tyramine SCHEMBL4111 0.97 TAAR1 (1.00) TAAR1KDM4EADRA2ASLC6A2ALDH1A1
Tyramine SCHEMBL30831107 0.97 TAAR1 (1.00) TAAR1KDM4EADRA2ASLC6A2ALDH1A1
Tyramine SCHEMBL30831130 0.97 TAAR1 (1.00) TAAR1KDM4EADRA2ASLC6A2ALDH1A1
Tyramine SCHEMBL2121 0.95 TDP1 (1.00) TAAR1KDM4EADRA2ASLC6A2ALDH1A1
Tyramine SCHEMBL31738431 0.95 TAAR1 (0.95) TAAR1KDM4EADRA2ASLC6A2ALDH1A1
Tyramine SCHEMBL7742928 0.95 TAAR1 (0.95) TAAR1KDM4EADRA2ASLC6A2ALDH1A1
Tyramine SCHEMBL32663617 0.95 TDP1 (1.00) TAAR1KDM4EADRA2ASLC6A2ALDH1A1
Tyramine SCHEMBL31718804 0.95 TAAR1 (0.95) TAAR1KDM4EADRA2ASLC6A2ALDH1A1
Tyramine SCHEMBL3950268 0.95 TAAR1 (0.95) TAAR1KDM4EADRA2ASLC6A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024108195-A1 COMBINATIONS OF MONOAMINE OXIDASE INHIBITORS AND SEROTONIN RECEPTOR AGONISTS AND THEIR THERAPEUTIC USE REMEDI, INC. (US) 2024-05-23 WO disclosed
EP-4355865-A1 NEW MICROBIAL DIAMINE OXIDASE DERIVED FROM YARROWIA LIPOLYTICA FOR THE DEGRADATION OF BIOGENIC AMINES Universität Hohenheim (DE) 2024-04-24 EP disclosed
CN-117904064-A Multi-copper oxidase of degradable biogenic amine from lactobacillus johnsonii and application thereof 江南大学 2024-04-19 CN disclosed
CN-117897478-A Novel microbial diamine oxidase derived from yarrowia lipolytica for biogenic amine degradation 霍恩海姆大学 2024-04-16 CN disclosed
EP-3067069-B1 HYDROGELS BASED ON POLYMERS OF DEXTRAN TYRAMINE AND TYRAMINE CONJUGATES OF NATURAL POLYMERS HY2CARE B V (NL) 2023-07-26 EP disclosed
WO-2022263031-A1 NEW MICROBIAL DIAMINE OXIDASE DERIVED FROM YARROWIA LIPOLYTICA FOR THE DEGRADATION OF BIOGENIC AMINES UNIVERSITÄT HOHENHEIM (DE) 2022-12-22 WO disclosed
EP-4105323-A1 NEW MICROBIAL DIAMINE OXIDASE DERIVED FROM YARROWIA LIPOLYTICA FOR THE DEGRADATION OF BIOGENIC AMINES Universität Hohenheim (DE) 2022-12-21 EP disclosed
CN-109810980-B Nucleic acid aptamer for specifically recognizing tyramine and application thereof 江南大学 2022-09-16 CN disclosed
CN-109810980-B Nucleic acid aptamer for specifically recognizing tyramine and application thereof 江南大学 2022-09-16 CN disclosed
US-20220175856-A1 UNRAVELING RECEPTOR-METABOLITE INTERACTIONS IN THE HUMAN MICROBIOME UNIV ROCKEFELLER (US) 2022-06-09 US disclosed
EP-2498824-B1 HYDROGELS BASED ON POLYMERS OF DEXTRAN TYRAMINE AND TYRAMINE CONJUGATES OF NATURAL POLYMERS UNIV TWENTE INST FOR BIOMEDICAL TECHNOLOGY AND TECHNICAL MEDICINE MIRA (NL) 2016-04-20 EP disclosed
CN-105399639-A Tyramine artificial antigen and antibody, and preparation methods and application thereof UNIV TIANJIN SCIENCE & TECH 2016-03-16 CN disclosed
US-9132201-B2 Hydrogels based on polymers of dextran tyramine and tyramine conjugates of natural polymers UNIVERSITY OF TWENTE, INSTITUTE FOR BIOMEDICAL AND TECHNICAL MEDICINE (MIRA) (NL) 2015-09-15 US disclosed
US-20120276069-A1 HYDROGELS BASED ON POLYMERS OF DEXTRAN TYRAMINE AND TYRAMINE CONJUGATES OF NATURAL POLYMERS HY2CARE B.V. (NL) 2012-11-01 US disclosed
EP-2498824-A2 HYDROGELS BASED ON POLYMERS OF DEXTRAN TYRAMINE AND TYRAMINE CONJUGATES OF NATURAL POLYMERS University of Twente, Institute for Biomedical Technology and Technical Medicine (MIRA) (NL) 2012-09-19 EP disclosed
WO-2011059326-A2 HYDROGELS BASED ON POLYMERS OF DEXTRAN TYRAMINE AND TYRAMINE CONJUGATES OF NATURAL POLYMERS UNIVERSITY OF TWENTE, INSTITUTE FOR BIOMEDICAL TECHNOLOGY AND TECHNICAL MEDICINE (MIRA) (NL) 2011-05-19 WO disclosed
US-20100143990-A1 FERMENTATIVE PRODUCTION OF HYDROXYTYROSOL DSM IP ASSETS B.V. (NL) 2010-06-10 US disclosed
US-20100068775-A1 NOVEL GENES FOR THE FERMENTATIVE PRODUCTION OF HYDROXYTYROSOL DSM IP ASSETS B.V. (NL) 2010-03-18 US disclosed
WO-2008064835-A1 FERMENTATIVE PRODUCTION OF HYDROXYTYROSOL DSM IP ASSETS B.V. (NL) 2008-06-05 WO disclosed
WO-2008064837-A2 NOVEL GENES FOR THE FERMENTATIVE PRODUCTION OF HYDROXYTYROSOL DSM IP ASSETS B.V. (NL) 2008-06-05 WO disclosed