SCHEMBL1807901

SCHEMBL1807901

CCCCOC(=O)N1CCC(=O)C(c2ccc(O[Si](C)(C)C(C)(C)C)cc2C)C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SMYD3 Q9H7B4 1/20 0.34
PLA2G2A P14555 2/20 0.33
HRH2 P25021 2/20 0.33
HRH1 P35367 2/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.32
KMT2A Q03164 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
MIF P14174 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
P2RY12 Q9H244 3/20 0.32
MMP13 P45452 1/20 0.32
CA12 O43570 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11898578 0.86 GPR119 (0.38) HSP90AA1HSP90AB1KDM4EALDH1A1CA12
SCHEMBL1804229 0.85 CA12 (0.36) HSP90AA1HSP90AB1CA12CA1CA9
SCHEMBL15166573 0.69 LMNA (0.48) LMNAPOLBSMN1; SMN2SMYD3HRH2
SCHEMBL30598434 0.69 NPC1 (0.46) LMNAPOLBSMN1; SMN2HRH2HRH1
SCHEMBL556212 0.69 MMP1 (0.37) MMP13CA12CA1CA9
SCHEMBL557260 0.69 ESR2 (0.51) KMT2AKDM4E
SCHEMBL29598912 0.68 LMNA (0.49) LMNAPOLBSMN1; SMN2SMYD3HRH2
SCHEMBL5156097 0.68 NR1H2 (0.41) SMN1; SMN2KMT2AKDM4E
SCHEMBL1445031 0.67 LMNA (0.48) LMNAPOLBSMN1; SMN2SMYD3PLA2G2A
SCHEMBL10097950 0.67 LMNA (0.48) LMNAPOLBSMN1; SMN2SMYD3HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488530-A1 SPIROCYCLIC PIPERIDINE DERIVATIVES USEFUL AS RENIN INHIBITORS Merck Canada Inc. (CA) 2012-08-22 EP disclosed
WO-2011057382-A1 SPIROCYCLIC PIPERIDINE DERIVATIVES USEFUL AS RENIN INHIBITORS MERCK FROSST CANADA LTD. (CA) 2011-05-19 WO disclosed