SCHEMBL18083000

SCHEMBL18083000

Cc1ccc2nc(C)c(C)nc2c1[N+](=O)[O-]

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
MAPT P10636 3/20 0.50
TDP1 Q9NUW8 3/20 0.47
TSHR P16473 4/20 0.46
MEN1 O00255 6/20 0.39
KMT2A Q03164 6/20 0.39
CYP3A4 P08684 1/20 0.38
NPBWR1 P48145 1/20 0.38
USP2 O75604 2/20 0.36
KEAP1 Q14145 2/20 0.36
NFE2L2 Q16236 2/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
POLB P06746 2/20 0.35
KDM4E B2RXH2 1/20 0.35
PKM P14618 1/20 0.35
APEX1 P27695 1/20 0.35
RECQL P46063 1/20 0.35
BLM P54132 1/20 0.35
CASP7 P55210 1/20 0.35
CASP6 P55212 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12964186 0.83 MEN1 (0.55) ALDH1A1MAPTTDP1TSHRMEN1
SCHEMBL18083002 0.82 KMT2A (0.49) ALDH1A1MAPTTDP1TSHRMEN1
SCHEMBL18083013 0.78 ALDH1A1 (0.58) ALDH1A1TDP1TSHRMEN1KMT2A
SCHEMBL27432919 0.76 ALDH1A1 (0.48) ALDH1A1TDP1TSHRMEN1KMT2A
SCHEMBL18083010 0.75 MEN1 (0.68) ALDH1A1MAPTTDP1TSHRMEN1
SCHEMBL5707397 0.74 MAPT (0.65) ALDH1A1MAPTTDP1TSHRMEN1
SCHEMBL4427648 0.73 ALDH1A1 (0.71) ALDH1A1TDP1TSHRCYP3A4SMN1; SMN2
SCHEMBL10390684 0.71 MEN1 (0.59) ALDH1A1MAPTTDP1TSHRMEN1
SCHEMBL11202171 0.71 MAPT (0.62) ALDH1A1MAPTTDP1CYP3A4SMN1; SMN2
SCHEMBL1225832 0.70 ALDH1A1 (1.00) ALDH1A1MAPTTDP1TSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9434701-B2 Aminoquinoxaline derivatives for treatment of neurodegenerative diseases CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2016-09-06 US disclosed